Target Details
| UniProt AC | Q9H2K2 |
|---|---|
| Gene Symbol | TNKS2 |
| Protein Name | Poly [ADP-ribose] polymerase tankyrase-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF13637 (Ank_4) PF00644 (PARP) PF07647 (SAM_2) |
Summary
- Multi-target molecules 746
- Clinical molecules 2
- Avg pChEMBL 7.83
Active Molecules (746)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SVDUOSYBBYZAAB
|
7.8 | IC50 | 2 | — | |
UEGWFDZLXJTQDG
|
7.8 | IC50 | 2 | — | |
UTGVEYXWHNPJKF
|
7.8 | IC50 | 3 | — | |
WWOMDTSWLDXWQW
|
7.8 | IC50 | 2 | — | |
ZBRBBDJXHBEGHX
|
7.8 | IC50 | 2 | — | |
ZGHNBPCNVXEKGL
|
7.8 | IC50 | 2 | — | |
ZHQHQOFGNSFGMK
|
7.8 | IC50 | 2 | — | |
HXVFMRKSTGSLPO
|
7.8 | IC50 | 2 | — | |
IFOOEZCGGVWMDI
|
7.8 | IC50 | 3 | — | |
KJYQLKOWSQIIBB
|
7.8 | IC50 | 2 | — | |
PERWUJINIMBCAY
|
7.8 | IC50 | 2 | — | |
QONNTUSBURAFST
|
7.8 | IC50 | 4 | — | |
QOUNQNYSBYTMLY
|
7.8 | IC50 | 2 | — | |
QWYIBGOLIBASGM
|
7.8 | IC50 | 2 | — | |
XSXNSAZKDIVZTL
|
7.8 | IC50 | 2 | — | |
ZGDNFPWQEQSQAA
|
7.8 | IC50 | 3 | — | |
ZZSBPGIGIUFJRA
|
7.8 | Kd | 46 | — | |
BDGRZWISYNXFKD
|
7.8 | IC50 | 3 | — | |
KXXRGTYOVUETBV
|
7.8 | IC50 | 3 | — | |
OUWQQYPQZGBQTQ
|
7.8 | IC50 | 2 | — | |
DKMQJZZVSIJOOY
|
7.8 | IC50 | 2 | — | |
DVRLXVRVRZISDR
|
7.8 | IC50 | 2 | — | |
FAAVFGPJNCDFEN
|
7.8 | IC50 | 2 | — | |
JAQISDRQXHHOJS
|
7.8 | IC50 | 2 | — | |
JDRRUNIVJVAXBH
|
7.8 | IC50 | 3 | — | |
JVUGYXTVNFUHII
|
7.8 | IC50 | 2 | — | |
KFHSJMVNDVHQGS
|
7.8 | IC50 | 2 | — | |
OMOFVXXXQGHNIN
|
7.8 | IC50 | 2 | — | |
PADREXIRIZBNMQ
|
7.8 | IC50 | 2 | — | |
WTVLTJMRTHFMJP
|
7.8 | IC50 | 2 | — | |
CWSRZPPZHBSBKK
|
7.8 | IC50 | 2 | — | |
DTOVAHAAYGWZJC
|
7.8 | IC50 | 2 | — | |
GNQUPDFWLAMRMB
|
7.8 | IC50 | 2 | — | |
APADCINNEFMGCF
|
7.8 | IC50 | 3 | — | |
DDIZJESACWEABB
|
7.8 | IC50 | 2 | — | |
GVSKTDUUGXDISO
|
7.8 | IC50 | 2 | — | |
IMXDGAQYSOUZNJ
|
7.8 | IC50 | 2 | — | |
XYPZDGAOLUTGCF
|
7.8 | IC50 | 2 | — | |
DWXBRPPQEBUSHN
|
7.8 | IC50 | 2 | — | |
HETQFLWNGHJHJZ
|
7.8 | IC50 | 2 | — | |
OMPYCYLPJBIPKG
|
7.8 | IC50 | 2 | — | |
GAIPKACDULOVTC
|
7.8 | IC50 | 3 | — | |
GXCGSCMUTWIBEU
|
7.8 | IC50 | 3 | — | |
FMURKSCWRQGCFO
|
7.7 | IC50 | 2 | — | |
GEXLAFHLVYHZAG
|
7.7 | IC50 | 2 | — | |
JLLCVKKYSDGUPY
|
7.7 | IC50 | 2 | — | |
QDPSTTBVXGPQGX
|
7.7 | IC50 | 2 | — | |
SRVUVWKCPPRJQZ
|
7.7 | IC50 | 2 | — | |
XGTNOTWEBRRAKO
|
7.7 | IC50 | 2 | — | |
YVWYZVHKYSEWDY
|
7.7 | IC50 | 2 | — |