Target Details
| UniProt AC | Q9H2K2 |
|---|---|
| Gene Symbol | TNKS2 |
| Protein Name | Poly [ADP-ribose] polymerase tankyrase-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF13637 (Ank_4) PF00644 (PARP) PF07647 (SAM_2) |
Summary
- Multi-target molecules 746
- Clinical molecules 2
- Avg pChEMBL 7.83
Active Molecules (746)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VFXBLJYICQUSGU
|
7.9 | IC50 | 2 | — | |
VLKQIEMXMFAOES
|
7.9 | IC50 | 2 | — | |
FOMOQTCFXCTELV
|
7.9 | IC50 | 2 | — | |
IGKALBMMBUOLAY
|
7.9 | IC50 | 2 | — | |
BMZFSQDDGKZEHW
|
7.9 | IC50 | 3 | — | |
FZQYCOUBRJEYBC
|
7.9 | IC50 | 2 | — | |
HANJAZOKICPNAX
|
7.9 | IC50 | 3 | — | |
HTLUBFSSIMOABR
|
7.9 | IC50 | 3 | — | |
ITFXLHSJWDBGLD
|
7.9 | IC50 | 2 | — | |
JJHZDQRUCBOSIK
|
7.9 | IC50 | 3 | — | |
KBFBQODMTQIXEB
|
7.9 | IC50 | 3 | — | |
MMWOCAKTGVKRBA
|
7.9 | IC50 | 2 | — | |
ODDUCZHVBOGEBZ
|
7.9 | IC50 | 2 | — | |
SJXSPWSYROZIMI
|
7.9 | IC50 | 2 | — | |
ULCIOMUEHZHNQU
|
7.9 | IC50 | 2 | — | |
WDZBHMSPANOWRC
|
7.9 | IC50 | 2 | — | |
WFJABTXVQUHYJP
|
7.9 | IC50 | 3 | — | |
ZQAMFUHPGNZLHA
|
7.9 | IC50 | 3 | — | |
KCPHCJUACXXHDI
|
7.9 | IC50 | 2 | — | |
STSCRAGBCYODMY
|
7.9 | IC50 | 8 | — | |
WZAAURATTBNWBC
|
7.9 | IC50 | 2 | — | |
BCVWBJPQPDBXMM
|
7.9 | IC50 | 3 | — | |
HWSBIYJZGFCBGQ
|
7.9 | IC50 | 2 | — | |
SMUYIABTVDLDHO
|
7.9 | IC50 | 2 | — | |
WLVFPFBPOHXOMK
|
7.9 | IC50 | 2 | — | |
XMLTXFYPZQGCBX
|
7.9 | IC50 | 2 | — | |
YIGLQGYCCCNBJG
|
7.9 | IC50 | 3 | — | |
ACORHZMZJPXEAA
|
7.9 | IC50 | 2 | — | |
DUYFEUQQISPFMM
|
7.9 | IC50 | 2 | — | |
FVSMOECHMBICED
|
7.9 | IC50 | 3 | — | |
PRPXVBJXNFAFSR
|
7.9 | IC50 | 2 | — | |
QSAWMHWYVIPNBM
|
7.9 | IC50 | 2 | — | |
QSAWMHWYVIPNBM
|
7.9 | IC50 | 2 | — | |
RJIONECKTUPQGG
|
7.9 | IC50 | 2 | — | |
RXVFAGGDYGCELS
|
7.9 | IC50 | 2 | — | |
XAQYIMOAZYNCLU
|
7.9 | IC50 | 2 | — | |
ZNLWDFKEMBITLP
|
7.9 | IC50 | 2 | — | |
RZFVLEJOHSLEFR
|
7.9 | IC50 | 4 | — | |
VUDVJHSDJGLCGJ
|
7.9 | IC50 | 2 | — | |
WAYVCDVUNSIWJI
|
7.9 | IC50 | 2 | — | |
CCMLHPSWIFWPCV
|
7.8 | IC50 | 2 | — | |
CLMCMCIANXSSCI
|
7.8 | IC50 | 2 | — | |
CVRMLBHUCXVUNB
|
7.8 | IC50 | 2 | — | |
GDPXXNADTSHZLW
|
7.8 | IC50 | 2 | — | |
HGMPUSYAOCCRQP
|
7.8 | IC50 | 3 | — | |
IKSANVUXVVKHGR
|
7.8 | IC50 | 2 | — | |
ILBZVTXOJSVUIM
|
7.8 | IC50 | 2 | — | |
JAQKAGMLMPVHSU
|
7.8 | IC50 | 2 | — | |
PBOOUBWKFXDCRA
|
7.8 | IC50 | 3 | — | |
RXWZXVGCPOUNQT
|
7.8 | IC50 | 3 | — |