Target Details
| UniProt AC | Q9H2K2 |
|---|---|
| Gene Symbol | TNKS2 |
| Protein Name | Poly [ADP-ribose] polymerase tankyrase-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF13637 (Ank_4) PF00644 (PARP) PF07647 (SAM_2) |
Summary
- Multi-target molecules 746
- Clinical molecules 2
- Avg pChEMBL 7.83
Active Molecules (746)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HIXCMHOBVDTAIE
|
8.1 | IC50 | 2 | — | |
IZGNMSCICRBUAB
|
8.1 | IC50 | 3 | — | |
MCMCBDOVNWSRNM
|
8.1 | IC50 | 2 | — | |
QDFBKHZKWYRNJE
|
8.1 | IC50 | 2 | — | |
SUKHPNUTRMBUST
|
8.1 | IC50 | 4 | — | |
BTVYOOANNCDQKM
|
8.1 | IC50 | 2 | — | |
FSNRYQUQAYKAPH
|
8.1 | IC50 | 4 | — | |
HIVDAZHBOHYAOK
|
8.1 | IC50 | 2 | — | |
MPGRGIIZXCNTKV
|
8.1 | IC50 | 2 | — | |
OUQKWLCWNMVJML
|
8.1 | IC50 | 2 | — | |
TXRJABUPPZKCNT
|
8.1 | IC50 | 2 | — | |
UVPFWJCKEJKCCW
|
8.1 | IC50 | 2 | — | |
XPFCXDCYIAOOBE
|
8.1 | IC50 | 2 | — | |
PAMGRUFJDHRZSY
|
8.1 | IC50 | 2 | — | |
XTWGYPAWWDNGTC
|
8.1 | IC50 | 3 | — | |
BSFWBIWYONWUDM
|
8.1 | IC50 | 2 | — | |
FXPQKIUFVMHDMQ
|
8.1 | IC50 | 2 | — | |
AANAXNPTHMWCLV
|
8.1 | IC50 | 2 | — | |
BCSYLIBZTSVMJI
|
8.1 | IC50 | 3 | — | |
MWUSNBQNIIMQRN
|
8.1 | IC50 | 4 | — | |
NFZIFTVDVOZOII
|
8.1 | IC50 | 2 | — | |
QTABKBZRAZXDQK
|
8.1 | IC50 | 2 | — | |
DBNHRWOXIIAGGS
|
8.1 | IC50 | 2 | — | |
GNNYYUFPAQKZRD
|
8.1 | IC50 | 2 | — | |
QOUNQNYSBYTMLY
|
8.1 | IC50 | 2 | — | |
RKIQHTHWSKPSAF
|
8.1 | IC50 | 2 | — | |
WPCRHWQMOWNQPY
|
8.1 | IC50 | 2 | — | |
UKLOIUCBRFPROX
|
8.0 | IC50 | 2 | — | |
OAXRVCSFISVGCI
|
8.0 | IC50 | 3 | — | |
OTGSIWARTZTTNU
|
8.0 | IC50 | 2 | — | |
QWYIBGOLIBASGM
|
8.0 | IC50 | 2 | — | |
WVGLSASLDWFLFS
|
8.0 | IC50 | 2 | — | |
GDPZGQDEZJRADO
|
8.0 | IC50 | 2 | — | |
GXKPLMIZTNQPMI
|
8.0 | IC50 | 2 | — | |
KGBRRRXNQADTEZ
|
8.0 | IC50 | 2 | — | |
KKBZHPTWKNTEDP
|
8.0 | IC50 | 2 | — | |
NEUUVLLFIFUTLB
|
8.0 | IC50 | 2 | — | |
DYSYSZSIEJMTPV
|
8.0 | IC50 | 2 | — | |
KXVJOZBQCTUYNT
|
8.0 | IC50 | 2 | — | |
IEJZGHYRQZYUPZ
|
8.0 | IC50 | 2 | — | |
HBRPUCMYDQNVOS
|
8.0 | IC50 | 3 | — | |
HRUWZYLXSAQFEL
|
8.0 | IC50 | 2 | — | |
MFVKIQGUHZYYOF
|
8.0 | IC50 | 2 | — | |
ZBJVKCDYVCVOIF
|
8.0 | IC50 | 3 | — | |
AMYVNCAWBFVJCR
|
8.0 | IC50 | 2 | — | |
CCVBOAMGJQRBBT
|
8.0 | IC50 | 3 | — | |
FAANBVRTVUGZKM
|
8.0 | IC50 | 2 | — | |
KZUPFZKALLNBBV
|
8.0 | IC50 | 2 | — | |
ZNAKJYRBQMWNHT
|
8.0 | IC50 | 2 | — | |
DBBRJAYFAWANIO
|
7.9 | IC50 | 2 | — |