Target Details
| UniProt AC | Q9H2K2 |
|---|---|
| Gene Symbol | TNKS2 |
| Protein Name | Poly [ADP-ribose] polymerase tankyrase-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF13637 (Ank_4) PF00644 (PARP) PF07647 (SAM_2) |
Summary
- Multi-target molecules 746
- Clinical molecules 2
- Avg pChEMBL 7.83
Active Molecules (746)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DGBBDMXUPJSMJV
|
8.6 | IC50 | 2 | — | |
MKFFPXHRRSVHGY
|
8.6 | IC50 | 2 | — | |
BPRGXQTYABGOBA
|
8.5 | IC50 | 3 | — | |
HDYMAMWGPQYCJR
|
8.5 | IC50 | 2 | — | |
BVCFVQGPDDYTEY
|
8.5 | IC50 | 2 | — | |
CEPPOYASQJVNOB
|
8.5 | IC50 | 2 | — | |
DJNXWSQAIXTYAO
|
8.5 | IC50 | 2 | — | |
GNQFITKNHVZOAH
|
8.5 | IC50 | 2 | — | |
NIPIEXNSQBQPML
|
8.5 | IC50 | 2 | — | |
ZPTIGCVQFHKQDB
|
8.5 | IC50 | 3 | — | |
MAISEOAFNXIHQI
|
8.5 | IC50 | 2 | — | |
JUVVMZKFNZPQIT
|
8.5 | IC50 | 3 | — | |
VWKAKGXPHIJGPD
|
8.5 | IC50 | 3 | — | |
YTZCTEISEKPJTQ
|
8.5 | IC50 | 3 | — | |
OCRURQUHABYGMH
|
8.5 | IC50 | 2 | — | |
RFMIZKCQNUDSTO
|
8.5 | IC50 | 3 | — | |
UXHCWVAWIZVATP
|
8.5 | IC50 | 2 | — | |
VJGJUSYNOCTGBZ
|
8.5 | IC50 | 2 | — | |
AXLLIVDKOSPBTM
|
8.5 | IC50 | 3 | — | |
PQOYFQLZYDRHBS
|
8.5 | IC50 | 2 | — | |
PSUPASCETWCMMJ
|
8.5 | IC50 | 2 | — | |
OKVSYWJACIIIKC
|
8.5 | IC50 | 2 | — | |
ZFHIMDPSSCABJV
|
8.5 | IC50 | 2 | — | |
NHVRXWDQNHZJTK
|
8.4 | IC50 | 3 | — | |
PAMUWGVDNNJVJY
|
8.4 | IC50 | 2 | — | |
YWNDUCFQXOXSHW
|
8.4 | IC50 | 2 | — | |
NLGGKDGPDAYIFS
|
8.4 | IC50 | 2 | — | |
AONMVAKCMAYUDD
|
8.4 | IC50 | 2 | — | |
CEKWANGMSIIGAG
|
8.4 | IC50 | 3 | — | |
XIFIENIKEZUQQD
|
8.4 | IC50 | 2 | — | |
DZBLVRUGYZNTPK
|
8.4 | IC50 | 2 | — | |
HMUTYRXLOPTZOV
|
8.4 | IC50 | 2 | — | |
UHPJRQMZYNOZHL
|
8.4 | IC50 | 2 | — | |
VKSDILZMXGBZJR
|
8.4 | IC50 | 3 | — | |
WOPOPFZLTYYWDV
|
8.4 | IC50 | 2 | — | |
IOMJPRIMVDNEHH
|
8.4 | IC50 | 2 | — | |
JLVRTMBMCWYGAL
|
8.4 | IC50 | 7 | — | |
KEKRVUGHUCXWSM
|
8.4 | IC50 | 2 | — | |
QWQWNLQBJNFADI
|
8.4 | IC50 | 2 | — | |
AFEVCFCEYWOQKD
|
8.4 | IC50 | 2 | — | |
ASRXCLRFDVRXIO
|
8.4 | IC50 | 2 | — | |
VQDCXZLOFBIDTL
|
8.4 | IC50 | 2 | — | |
FUQQJIVTKMJOTI
|
8.4 | IC50 | 2 | — | |
HSKIFVPMPRQUPP
|
8.3 | IC50 | 2 | — | |
HXWKRLPCYVNDNE
|
8.3 | IC50 | 2 | — | |
GMZHCIWODQRBEX
|
8.3 | IC50 | 2 | — | |
IHBILSNANZVSHM
|
8.3 | IC50 | 2 | — | |
KBKQSDRVJSIUST
|
8.3 | IC50 | 2 | — | |
KVVODYVRKLLEIQ
|
8.3 | IC50 | 2 | — | |
MILMCUZGEDRYHA
|
8.3 | IC50 | 3 | — |