Target Details
| UniProt AC | Q9H2K2 |
|---|---|
| Gene Symbol | TNKS2 |
| Protein Name | Poly [ADP-ribose] polymerase tankyrase-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF13637 (Ank_4) PF00644 (PARP) PF07647 (SAM_2) |
Summary
- Multi-target molecules 746
- Clinical molecules 2
- Avg pChEMBL 7.83
Active Molecules (746)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FWEQRPGVBGGLAV
|
8.9 | IC50 | 2 | — | |
ZRQMVNYALKQFAB
|
8.9 | IC50 | 3 | — | |
KRJJSTRNPUSJST
|
8.9 | IC50 | 2 | — | |
RKTAKASHRFDDHH
|
8.9 | IC50 | 2 | — | |
ZTIZYNDBJGONBV
|
8.9 | IC50 | 2 | — | |
YKDCXYUWCYJSJW
|
8.9 | IC50 | 2 | — | |
GWBSSUZALYDTAX
|
8.8 | IC50 | 3 | — | |
HBJBOCIRHMWTFT
|
8.8 | IC50 | 3 | — | |
IFGZJOCKQVPMQP
|
8.8 | IC50 | 3 | — | |
VJHDAFXRSRJKPL
|
8.8 | IC50 | 3 | — | |
ZJHLKLRWORVGKO
|
8.8 | IC50 | 3 | — | |
JPLMWQFVSFXHLA
|
8.8 | IC50 | 2 | — | |
SSRCPYMXFHISQW
|
8.8 | IC50 | 3 | — | |
WDAVNQKSHQVPKD
|
8.8 | IC50 | 4 | — | |
AOMPHWKJTUPEOB
|
8.8 | IC50 | 3 | — | |
FZJXZJRCQJPQDJ
|
8.8 | IC50 | 2 | — | |
SRMMCJRPCQBABR
|
8.8 | IC50 | 3 | — | |
ZDXHDNKNNXPLHR
|
8.8 | IC50 | 2 | — | |
GWKQMSZYRPKGIR
|
8.7 | IC50 | 3 | — | |
HEJKSHFADGJFLY
|
8.7 | IC50 | 2 | — | |
JXORYUCIOICGOX
|
8.7 | IC50 | 3 | — | |
PPGDXAFAEKIBAL
|
8.7 | IC50 | 3 | — | |
XBMLIULZOSKFDL
|
8.7 | IC50 | 2 | — | |
ARCOJIXZDJYBCH
|
8.7 | IC50 | 2 | — | |
QXYNHQXOVDACBV
|
8.7 | IC50 | 2 | — | |
ANMLHQJBUZSTOM
|
8.7 | IC50 | 2 | — | |
AOMPHWKJTUPEOB
|
8.7 | IC50 | 3 | — | |
DYMJRWLCTOEALR
|
8.7 | IC50 | 2 | — | |
KVBKYZXBOMQZDK
|
8.7 | IC50 | 2 | — | |
WWKKOAKRYQQEBT
|
8.7 | IC50 | 3 | — | |
BGJRUZLMBXELSD
|
8.7 | IC50 | 3 | — | |
PCRNXFSEUXATPP
|
8.7 | IC50 | 2 | — | |
SRAYYDCMTKRHDU
|
8.7 | IC50 | 2 | — | |
UQSSCRPZDDBPIX
|
8.7 | IC50 | 3 | — | |
IQJONQOJCNHAQX
|
8.7 | IC50 | 2 | — | |
ITIZYYXRCNBXRH
|
8.7 | IC50 | 2 | — | |
PEOXTCZVHIZAKJ
|
8.7 | IC50 | 2 | — | |
XTEDLLOZIRDMGM
|
8.7 | IC50 | 3 | — | |
BDBCLQYLIMPBKR
|
8.6 | IC50 | 2 | — | |
NOMOJZWMCUJGHN
|
8.6 | IC50 | 3 | — | |
NZVGSVJJAPFBDQ
|
8.6 | IC50 | 2 | — | |
YJZCHZMPLVJNHG
|
8.6 | IC50 | 2 | — | |
ZBQDZIKGERQLAW
|
8.6 | IC50 | 2 | — | |
DJQNMMNQHCULEE
|
8.6 | IC50 | 2 | — | |
IKPHQSQQUCQZBC
|
8.6 | IC50 | 2 | — | |
WQPAUZHGHHSUOT
|
8.6 | IC50 | 3 | — | |
YTDAPYITALQSLF
|
8.6 | IC50 | 2 | — | |
BVBKPRYPLQAWKE
|
8.6 | IC50 | 3 | — | |
SFJDBLUTKNOEFD
|
8.6 | IC50 | 2 | — | |
VNDAUZPOPZSKLR
|
8.6 | IC50 | 2 | — |