Target Details
| UniProt AC | Q9H2K2 |
|---|---|
| Gene Symbol | TNKS2 |
| Protein Name | Poly [ADP-ribose] polymerase tankyrase-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF13637 (Ank_4) PF00644 (PARP) PF07647 (SAM_2) |
Summary
- Multi-target molecules 746
- Clinical molecules 2
- Avg pChEMBL 7.83
Active Molecules (746)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QZHUFUOXNJRYML
|
9.4 | IC50 | 4 | — | |
FUQQJIVTKMJOTI
|
9.3 | IC50 | 2 | — | |
LPJHLUNKDITEKL
|
9.3 | IC50 | 2 | — | |
ORMXFDLXICVSQJ
|
9.3 | IC50 | 2 | — | |
TZBJUABBPHUUCL
|
9.3 | IC50 | 3 | — | |
CADYSKUZMAIDBU
|
9.3 | IC50 | 4 | — | |
SHCKGNRFHFRCLF
|
9.3 | IC50 | 3 | — | |
KCCHUDANIWRWFS
|
9.3 | IC50 | 3 | — | |
NUCKGGSDYMOWIS
|
9.3 | IC50 | 2 | — | |
CKOUULRCBKAWEI
|
9.3 | IC50 | 4 | — | |
FHWNIOZFSDHKSG
|
9.3 | IC50 | 4 | — | |
TXRJABUPPZKCNT
|
9.3 | IC50 | 2 | — | |
JKUCQWSEJQYAJC
|
9.3 | IC50 | 3 | — | |
BCSYLIBZTSVMJI
|
9.3 | IC50 | 3 | — | |
HBWPYEOAXUKSAJ
|
9.2 | IC50 | 2 | — | |
QFFQVTQVYJNUQK
|
9.2 | IC50 | 2 | — | |
TVAKNHJAERNITR
|
9.2 | IC50 | 2 | — | |
KCXFNUZJEYUGTK
|
9.2 | IC50 | 3 | — | |
KTIYJXKGHKLGEV
|
9.2 | IC50 | 3 | — | |
WCPTUQOMNJBIET
|
9.2 | IC50 | 3 | — | |
YSXKCOVMSIANLW
|
9.2 | IC50 | 2 | — | |
ZBQNBDDBQXSUCN
|
9.2 | IC50 | 2 | — | |
XHNQPDNRQBXYJO
|
9.2 | IC50 | 2 | — | |
ZJAQFWFBBDESAQ
|
9.2 | IC50 | 3 | — | |
DPLIWMOJVZZKPZ
|
9.2 | IC50 | 2 | — | |
MOMSZDNLTDTPMD
|
9.2 | IC50 | 3 | — | |
WQGFJZQGDWKRMN
|
9.2 | IC50 | 4 | — | |
AXAVZUGQTQESKM
|
9.2 | IC50 | 2 | — | |
QKUQIWILQMTNRG
|
9.2 | IC50 | 2 | — | |
NRGTYYQXOBIJNO
|
9.2 | IC50 | 3 | — | |
OOQHGTMJHBCFLX
|
9.1 | IC50 | 2 | — | |
PHWWAZGJHKJDLI
|
9.1 | IC50 | 2 | — | |
YFRRHPBZXLBANM
|
9.1 | IC50 | 3 | — | |
HKIWKJRHIASRSM
|
9.1 | IC50 | 3 | — | |
JWTZFQHEWRUOBW
|
9.1 | IC50 | 3 | — | |
OEHCCJHWIUUHFU
|
9.1 | IC50 | 3 | — | |
ARDLHSGXMZNXNJ
|
9.1 | IC50 | 2 | — | |
ZMDXCCGWVIFDMF
|
9.1 | IC50 | 2 | — | |
JDZQHCQYJAHSCQ
|
9.1 | IC50 | 3 | — | |
MPXAEYSGFKRDQM
|
9.1 | IC50 | 7 | — | |
MGEFDMCHHLACOB
|
9.0 | IC50 | 4 | — | |
APINASOTMBYJNI
|
9.0 | IC50 | 2 | — | |
JMPOHTPVCKISQL
|
9.0 | IC50 | 3 | — | |
MOMSZDNLTDTPMD
|
9.0 | IC50 | 2 | — | |
OIHAQLWXPNRBJG
|
9.0 | IC50 | 2 | — | |
SSRCPYMXFHISQW
|
9.0 | IC50 | 3 | — | |
UIPJAQKAZCQVPU
|
9.0 | IC50 | 3 | — | |
UXGMDGPWMVIMFP
|
9.0 | IC50 | 2 | — | |
WYQKLIGAUQKHIE
|
9.0 | IC50 | 3 | — | |
LBUVXBLWWXNUHN
|
9.0 | IC50 | 2 | — |