Target Details
| UniProt AC | Q9H2K2 |
|---|---|
| Gene Symbol | TNKS2 |
| Protein Name | Poly [ADP-ribose] polymerase tankyrase-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF13637 (Ank_4) PF00644 (PARP) PF07647 (SAM_2) |
Summary
- Multi-target molecules 746
- Clinical molecules 2
- Avg pChEMBL 7.83
Active Molecules (746)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZKKFHBDYTOSSFW
|
6.8 | IC50 | 2 | — | |
BWTOWBOMDHKCDB
|
6.8 | IC50 | 7 | — | |
FLCHMGRFSJQORK
|
6.8 | IC50 | 3 | — | |
GERFIVKNGYXTHK
|
6.8 | IC50 | 2 | — | |
RBDQSAKXGCRFGL
|
6.8 | IC50 | 2 | — | |
JFJGQBKALIOSDA
|
6.8 | IC50 | 3 | — | |
RLEBLHKNUCJVNF
|
6.8 | IC50 | 2 | — | |
DKYAMBSWXNVNIR
|
6.8 | IC50 | 2 | — | |
JKCKQJATUNERKN
|
6.8 | IC50 | 2 | — | |
CXANDIUMTJKCEI
|
6.8 | IC50 | 3 | — | |
ZKUPHCJCVQFXDM
|
6.8 | IC50 | 2 | — | |
ZMGPDWHTUMUFPT
|
6.8 | IC50 | 2 | — | |
AHJJFIGHBOPXKV
|
6.8 | IC50 | 2 | — | |
JRDFYUFZPYBDNH
|
6.7 | IC50 | 2 | — | |
WFUUHEFQQUZRTP
|
6.7 | IC50 | 2 | — | |
JXSWEIKYXMJGGG
|
6.7 | IC50 | 3 | — | |
REUQDXNRIHMJKE
|
6.7 | IC50 | 2 | — | |
DTMHAFMUJHYVGK
|
6.7 | IC50 | 3 | — | |
FKPMZNSEGYFIDN
|
6.7 | IC50 | 3 | — | |
HMZVOPJPTNTGGO
|
6.7 | IC50 | 2 | — | |
LUYWAGVRXKSNLL
|
6.7 | IC50 | 2 | — | |
OPHKKQQCOYMLPW
|
6.7 | IC50 | 3 | — | |
XNKSDYBDUSFGDT
|
6.7 | IC50 | 2 | — | |
ZDDPBFWHZOJFHF
|
6.7 | IC50 | 6 | — | |
AFXJUCILCGBUNX
|
6.7 | IC50 | 4 | — | |
IRYZTIMDNVDWKI
|
6.7 | IC50 | 2 | — | |
UVYVRAATXCFMQQ
|
6.7 | IC50 | 4 | — | |
XZTBVJZEZAGWMB
|
6.7 | IC50 | 3 | — | |
BVCFVQGPDDYTEY
|
6.7 | IC50 | 2 | — | |
HPVNLHNRECCVHK
|
6.7 | IC50 | 2 | — | |
MHQFEYXRRZRKBA
|
6.7 | IC50 | 3 | — | |
USJIPGUTADKMST
|
6.7 | IC50 | 2 | — | |
FNYTYXJFOSRUTI
|
6.7 | IC50 | 3 | — | |
QOUNQNYSBYTMLY
|
6.7 | IC50 | 2 | — | |
WPCRHWQMOWNQPY
|
6.7 | IC50 | 2 | — | |
BMPSOKZAIFFMLK
|
6.6 | IC50 | 6 | — | |
TWBVIDDSIBCAOI
|
6.6 | IC50 | 2 | — | |
PVUNOEJZLPVTPG
|
6.6 | IC50 | 2 | — | |
YZLWXJLWHXPUGR
|
6.6 | IC50 | 2 | — | |
QEFRLEQZTKAQJC
|
6.6 | IC50 | 2 | — | |
RNMBZYKZMPEIAZ
|
6.6 | IC50 | 2 | — | |
NKPDQKILCAOJCZ
|
6.6 | IC50 | 2 | — | |
OPXUZDOALWXAIC
|
6.6 | IC50 | 2 | — | |
VJWOVHIEGPXVQC
|
6.6 | IC50 | 2 | — | |
PAMHLAWFGRSETB
|
6.5 | IC50 | 2 | — | |
AQSATLITSNDZSM
|
6.5 | IC50 | 2 | — | |
BSGNOJZPCZALIF
|
6.5 | IC50 | 2 | — | |
ONWFSNLHAZAPLW
|
6.5 | IC50 | 3 | — | |
PVRVKAMGYYHFJO
|
6.5 | IC50 | 3 | — | |
ISZWRZGKEWQACU
|
6.5 | IC50 | 3 | — |