Target Details
| UniProt AC | Q9H2K2 |
|---|---|
| Gene Symbol | TNKS2 |
| Protein Name | Poly [ADP-ribose] polymerase tankyrase-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF13637 (Ank_4) PF00644 (PARP) PF07647 (SAM_2) |
Summary
- Multi-target molecules 746
- Clinical molecules 2
- Avg pChEMBL 7.83
Active Molecules (746)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CQDSSYSRDXRGLW
|
7.4 | IC50 | 2 | — | |
DXJNIJJCRJVJHJ
|
7.4 | IC50 | 2 | — | |
HOSHPNDTAUJRNF
|
7.4 | IC50 | 2 | — | |
IGFHGNCTXXHXTG
|
7.4 | IC50 | 2 | — | |
ISIFMYDJQDUUNJ
|
7.4 | IC50 | 2 | — | |
SGEGLEFCEAUJJJ
|
7.4 | IC50 | 2 | — | |
ZEQVKZNUMQSOLV
|
7.4 | IC50 | 2 | — | |
ZUBOEZVHUJULCK
|
7.4 | IC50 | 3 | — | |
CXHHTZQIOFCSNN
|
7.4 | IC50 | 2 | — | |
WLZJEOODSSBWMB
|
7.4 | IC50 | 3 | — | |
QOEFYUDGLXWPLV
|
7.4 | IC50 | 2 | — | |
GFUWRTZMZMICED
|
7.4 | IC50 | 3 | — | |
NGWLKFVMSQZGRO
|
7.4 | IC50 | 3 | — | |
NIDNWZWMIAQVNK
|
7.4 | IC50 | 2 | — | |
NQNHZFQNGJXOBP
|
7.4 | IC50 | 2 | — | |
QERGZXHGTSDAGX
|
7.4 | IC50 | 2 | — | |
WEVHGUILVANSPZ
|
7.4 | IC50 | 2 | — | |
ATLOZOFUVNDOGJ
|
7.4 | IC50 | 2 | — | |
FDWCAGLPVGJZGX
|
7.4 | IC50 | 3 | — | |
MCCQXQRJNJXHRG
|
7.4 | IC50 | 3 | — | |
ULCGWFIERYSNSV
|
7.4 | IC50 | 2 | — | |
WQQPDDQFWUCFDH
|
7.4 | IC50 | 2 | — | |
DDFLFKTXUWPNMV
|
7.3 | IC50 | 3 | — | |
DDFLFKTXUWPNMV
|
7.3 | IC50 | 3 | — | |
UYLLGWXNACFQPE
|
7.3 | IC50 | 2 | — | |
LNBBOOMVYRTUHU
|
7.3 | IC50 | 2 | — | |
QWKZXCNQEFMJAM
|
7.3 | IC50 | 3 | — | |
AXUQAIVLNXVOPO
|
7.3 | IC50 | 2 | — | |
HMPAJUGZRUZDQJ
|
7.3 | IC50 | 2 | — | |
JLFSBHQQXIAQEC
|
7.3 | IC50 | 4 | — | |
LDWBPQDBDYNXIG
|
7.3 | IC50 | 2 | — | |
OMOFVXXXQGHNIN
|
7.3 | IC50 | 2 | — | |
ZFSOEIOPMMKKQB
|
7.3 | IC50 | 2 | — | |
ZPLCRPBMZNZKDA
|
7.3 | IC50 | 2 | — | |
FASROOIKQQJQSJ
|
7.3 | IC50 | 2 | — | |
HYPDQYLAVWCCSO
|
7.3 | IC50 | 2 | — | |
DEGIMKQHUITSSN
|
7.3 | IC50 | 2 | — | |
HETSSARHFAGODR
|
7.3 | IC50 | 3 | — | |
JGLLGSHEXZAGLB
|
7.3 | IC50 | 2 | — | |
KKRQGICUYMCZFH
|
7.3 | IC50 | 2 | — | |
LTQNPKURAUAWPU
|
7.3 | IC50 | 2 | — | |
QFPKMPQXSRPUCK
|
7.3 | IC50 | 2 | — | |
RMPXVEDDRZOQIA
|
7.3 | IC50 | 2 | — | |
JLUWGYRKHZWQDW
|
7.3 | IC50 | 2 | — | |
YUZGATGNXIWEAT
|
7.3 | IC50 | 2 | — | |
OAXYPHWHZZNXGF
|
7.3 | IC50 | 2 | — | |
LCGPTLVHGJYCAG
|
7.2 | IC50 | 2 | — | |
ZGSXEXBYLJIOGF
|
7.2 | IC50 | 2 | — | |
ZWIJUUMFHSAWDX
|
7.2 | IC50 | 3 | — | |
IUHUYCJRJLWYHF
|
7.2 | IC50 | 2 | — |