Target Details
| UniProt AC | Q9H2K2 |
|---|---|
| Gene Symbol | TNKS2 |
| Protein Name | Poly [ADP-ribose] polymerase tankyrase-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF13637 (Ank_4) PF00644 (PARP) PF07647 (SAM_2) |
Summary
- Multi-target molecules 746
- Clinical molecules 2
- Avg pChEMBL 7.83
Active Molecules (746)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LKLUJAFKWQGZNH
|
10.1 | IC50 | 2 | — | |
CFKUCYZMLBDUOB
|
10.0 | IC50 | 2 | — | |
VADYPHREEXKWAX
|
10.0 | IC50 | 2 | — | |
MPQCBOWATMYRKR
|
9.8 | IC50 | 2 | — | |
ZWSDFCUUVVGTIL
|
9.8 | IC50 | 2 | — | |
GMBPALAESNNJFY
|
9.8 | IC50 | 2 | — | |
PSRZACYIKWDSNE
|
9.8 | IC50 | 2 | — | |
CSZYQIKNQBWYMC
|
9.7 | IC50 | 3 | — | |
MONJJZAAKCCXFC
|
9.7 | IC50 | 2 | — | |
PPFZSMPPXPFDAK
|
9.7 | IC50 | 2 | — | |
QXYNHQXOVDACBV
|
9.7 | IC50 | 2 | — | |
XSSGDRWJVHTQAM
|
9.7 | IC50 | 2 | — | |
FGJFFFXLPMJDRZ
|
9.7 | IC50 | 3 | — | |
NENMCAZABRSHBQ
|
9.7 | IC50 | 2 | — | |
HILQRGHXDPSDBM
|
9.7 | IC50 | 2 | — | |
KTIYJXKGHKLGEV
|
9.7 | IC50 | 3 | — | |
AFHDZWZQZNOEPI
|
9.7 | IC50 | 4 | — | |
SWIOCYMLKFHIEX
|
9.7 | IC50 | 2 | — | |
MKFFPXHRRSVHGY
|
9.7 | IC50 | 3 | — | |
AAGQBOZLMIXHHO
|
9.6 | IC50 | 3 | — | |
XXNXCOLKURBCKS
|
9.6 | IC50 | 2 | — | |
YFRRHPBZXLBANM
|
9.6 | IC50 | 2 | — | |
ZBYOHASAEQTYGT
|
9.6 | IC50 | 2 | — | |
ZJNATVSUTRSLJP
|
9.6 | IC50 | 3 | — | |
IIMAZMNSHUIJDI
|
9.6 | IC50 | 2 | — | |
HNNOUHLGNDSYMQ
|
9.6 | IC50 | 2 | — | |
JVPFBWSJCYHTIN
|
9.6 | IC50 | 3 | — | |
RGDWKTYYFMMDGT
|
9.6 | IC50 | 2 | — | |
LMUIMYHRSNNJLB
|
9.6 | IC50 | 2 | — | |
IGTMNQSNSCDFLH
|
9.5 | IC50 | 2 | — | |
BZWBNQLFSDLENC
|
9.5 | IC50 | 2 | — | |
RGSSADMOZOOPCT
|
9.5 | IC50 | 4 | — | |
AICJSAOJHVWPBE
|
9.5 | IC50 | 2 | — | |
FDICCIFLUUYDFS
|
9.5 | IC50 | 4 | — | |
RHCZTJJJLXGIDT
|
9.5 | IC50 | 4 | — | |
ZTMJFCMMULUTEL
|
9.5 | IC50 | 2 | — | |
MEQYFMGLIUJKRI
|
9.5 | IC50 | 2 | — | |
KCIAHAOBFVPQKW
|
9.5 | IC50 | 2 | — | |
ANHWOOWZYAWFMI
|
9.5 | IC50 | 2 | — | |
KPDGLOCQRBTKHT
|
9.5 | IC50 | 3 | — | |
CVEOMWCWJJWSAV
|
9.4 | IC50 | 2 | — | |
MAJDINHMZAHJEQ
|
9.4 | IC50 | 2 | — | |
JCXKRJIIGPWGFB
|
9.4 | IC50 | 2 | — | |
OFLAMXGZJOGJGE
|
9.4 | IC50 | 2 | — | |
ABCZORPRBCURRK
|
9.4 | IC50 | 3 | — | |
BTVYOOANNCDQKM
|
9.4 | IC50 | 2 | — | |
BGRUEOQGBAKLPG
|
9.4 | IC50 | 2 | — | |
VXCLLARJZBLHAR
|
9.4 | IC50 | 2 | — | |
NLHWNHOBNJGSMX
|
9.4 | IC50 | 3 | — | |
JWNWTMMYAWEEFL
|
9.4 | IC50 | 2 | — |