Target Details
| UniProt AC | Q9H1R3 |
|---|---|
| Gene Symbol | MYLK2 |
| Protein Name | Myosin light chain kinase 2, skeletal/cardiac muscle |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 22
- Clinical molecules 8
- Avg pChEMBL 6.55
KEGG Pathways (10)
Associated Diseases (1)
Active Molecules (22)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GCIKSSRWRFVXBI
|
7.4 | Kd | 109 | Yes | |
WINHZLLDWRZWRT
|
7.3 | Kd | 201 | Yes | |
YYLKKYCXAOBSRM
|
7.3 | Kd | 191 | — | |
UIARLYUEJFELEN
|
7.2 | Kd | 289 | Yes | |
HKSZLNNOFSGOKW
|
7.2 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
7.2 | Kd | 213 | — | |
PIQCTGMSNWUMAF
|
7.0 | Kd | 137 | Yes | |
CTNPALGJUAXMMC
|
6.7 | Kd | 151 | — | |
VAARYSWULJUGST
|
6.7 | Kd | 119 | Yes | |
ODPGGGTTYSGTGO
|
6.5 | Kd | 153 | — | |
RKBMAROJKLHAMI
|
6.5 | IC50 | 6 | — | |
HVHRHDHQHUAOQI
|
6.3 | IC50 | 5 | — | |
ZFXGOGALEGXWEL
|
6.2 | IC50 | 5 | — | |
ZVSNSFQQKSZZMY
|
6.2 | IC50 | 7 | — | |
SIXVRXARNAVBTC
|
6.2 | IC50 | 12 | — | |
OYONTEXKYJZFHA
|
6.0 | Kd | 69 | Yes | |
UCBIQZUJJSVQHL
|
6.0 | Kd | 8 | — | |
AAKJLRGGTJKAMG
|
6.0 | Kd | 50 | Yes | |
OUSFTKFNBAZUKL
|
6.0 | Kd | 58 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |