Target Details
| UniProt AC | Q9H0K1 |
|---|---|
| Gene Symbol | SIK2 |
| Protein Name | Serine/threonine-protein kinase SIK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF23312 (UBA_SIK3) |
Summary
- Multi-target molecules 250
- Clinical molecules 23
- Avg pChEMBL 7.83
KEGG Pathways (1)
Active Molecules (250)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IDHYGWPCQJKIOG
|
7.7 | IC50 | 3 | — | |
HWSYLCVSNZMWCP
|
7.6 | IC50 | 3 | — | |
PBBRWFOVCUAONR
|
7.6 | Ki | 26 | Yes | |
RGUMENUIWKKDQS
|
7.6 | IC50 | 3 | — | |
UGMDEPACJFWQTK
|
7.6 | IC50 | 3 | — | |
VAARYSWULJUGST
|
7.6 | Kd | 119 | Yes | |
RIJYZTZQMRSSEU
|
7.6 | IC50 | 3 | — | |
UBPYILGKFZZVDX
|
7.5 | Kd | 130 | Yes | |
LOLPPWBBNUVNQZ
|
7.5 | Kd | 97 | Yes | |
NELFAFAXIZFQJB
|
7.5 | IC50 | 3 | — | |
PMXGPFCKENCVOL
|
7.5 | IC50 | 3 | — | |
XPSCTAWDRZNUCF
|
7.5 | IC50 | 3 | — | |
WXBMZGPQDSOPBO
|
7.5 | IC50 | 2 | — | |
PJFVPKCPIJSWQT
|
7.5 | IC50 | 3 | — | |
JPMOTSGSTDSLFB
|
7.4 | IC50 | 2 | — | |
SZGFJHKSBCTFLK
|
7.4 | IC50 | 3 | — | |
VQINULODWGEVBB
|
7.4 | IC50 | 4 | — | |
ULGBXNOOIDGVSQ
|
7.4 | IC50 | 3 | — | |
YFVBBRRMTKZKEK
|
7.4 | IC50 | 2 | — | |
YFNWWNRZJGMDBR
|
7.3 | Kd | 35 | — | |
CSGQVNMSRKWUSH
|
7.3 | Kd | 21 | — | |
JXJARIRMZQINMV
|
7.3 | IC50 | 3 | — | |
QKNBRNSGPNCARD
|
7.3 | IC50 | 9 | — | |
XASOHFCUIQARJT
|
7.3 | IC50 | 4 | — | |
GLLIRMCFYAPERL
|
7.3 | IC50 | 2 | — | |
NCQKIKYQHVNIMN
|
7.3 | IC50 | 2 | — | |
UWLKLAVEUJFHNV
|
7.3 | IC50 | 3 | — | |
INDWAJWLSOYKGH
|
7.2 | IC50 | 3 | — | |
KOZFSFOOLUUIGY
|
7.2 | Kd | 88 | Yes | |
CRLZGLXSANQWFT
|
7.2 | IC50 | 6 | — | |
UKBGBACORPRCGG
|
7.2 | IC50 | 17 | — | |
DVQJNPZTPKFTFL
|
7.1 | IC50 | 3 | — | |
QAMUWRFOZKONDU
|
7.1 | IC50 | 7 | — | |
NHHQJBCNYHBUSI
|
7.1 | Kd | 220 | — | |
VCZDFACOFNRTMG
|
7.0 | IC50 | 6 | — | |
ZZSBPGIGIUFJRA
|
7.0 | Kd | 46 | — | |
JOOXLOJCABQBSG
|
7.0 | Kd | 139 | — | |
ANQJLVHORSBOEP
|
7.0 | IC50 | 3 | — | |
PIQCTGMSNWUMAF
|
7.0 | Ki | 137 | Yes | |
LEGLVJKJPHFNFK
|
7.0 | IC50 | 2 | — | |
WKDACQVEJIVHMZ
|
6.9 | Kd | 46 | — | |
ZMNVPNNTSQXNLO
|
6.9 | IC50 | 3 | — | |
RJLWSBWYWAAETQ
|
6.9 | IC50 | 3 | — | |
RTRHXDLGBINMNM
|
6.9 | IC50 | 5 | — | |
MGGBYMDAPCCKCT
|
6.9 | Kd | 23 | — | |
IEFFSHLHNYVSEF
|
6.9 | IC50 | 8 | — | |
TZEWBPGVTYPITP
|
6.9 | IC50 | 5 | — | |
QWACVNYZRLANPQ
|
6.9 | IC50 | 2 | — | |
INSVCYRFDCTMIA
|
6.9 | IC50 | 5 | — | |
DUDGRZRMJYRPNL
|
6.8 | IC50 | 2 | — |