Target Details
| UniProt AC | Q9H0K1 |
|---|---|
| Gene Symbol | SIK2 |
| Protein Name | Serine/threonine-protein kinase SIK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF23312 (UBA_SIK3) |
Summary
- Multi-target molecules 250
- Clinical molecules 23
- Avg pChEMBL 7.83
KEGG Pathways (1)
Active Molecules (250)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CBLISIIXOMPZFZ
|
8.2 | IC50 | 3 | — | |
HJHOVADSVUHROW
|
8.2 | IC50 | 3 | — | |
ZBNZXTGUTAYRHI
|
8.2 | Kd | 102 | Yes | |
PBQKEWXFKZOWAZ
|
8.2 | IC50 | 3 | — | |
IAYGCINLNONXHY
|
8.2 | Kd | 50 | — | |
ZHXIRQMWOVKZBZ
|
8.2 | IC50 | 2 | — | |
XCGUGTWHQADPNS
|
8.1 | IC50 | 3 | — | |
DWTXIQAMWBBKJO
|
8.1 | IC50 | 2 | — | |
CKVPYFIWJCSSSQ
|
8.1 | IC50 | 3 | — | |
KCUIXXONNLBRFH
|
8.1 | IC50 | 3 | — | |
UARVSLPFGRKWQN
|
8.1 | IC50 | 11 | — | |
YHKXOSIWOVIDSP
|
8.1 | IC50 | 3 | — | |
ZGIZZXHFELWYTH
|
8.1 | IC50 | 3 | — | |
ZBCMHWUFWQFPLV
|
8.1 | IC50 | 9 | — | |
SGMHSWUFNYQVBA
|
8.0 | IC50 | 9 | — | |
XIAKIYQZBHRETP
|
8.0 | IC50 | 3 | — | |
JDNFAAUUFUBZKC
|
8.0 | IC50 | 3 | — | |
MXJMJNRCJKHFPP
|
8.0 | IC50 | 10 | — | |
PBCZSGKMGDDXIJ
|
8.0 | Kd | 68 | Yes | |
RYYNGWLOYLRZLK
|
8.0 | Kd | 45 | — | |
HRKJFKJZUNJKNU
|
8.0 | IC50 | 10 | — | |
OHQUFRHYRLCLFC
|
7.9 | IC50 | 3 | — | |
ZLOMEKCROOJNIA
|
7.9 | IC50 | 2 | — | |
LZUYOYKXEXENTQ
|
7.9 | IC50 | 5 | — | |
OFIFLUFVENTCNZ
|
7.9 | IC50 | 11 | — | |
MYYIXDJCLRMEBI
|
7.9 | IC50 | 3 | — | |
DFZKXFCZKLBBRG
|
7.9 | IC50 | 3 | — | |
PKJTVQJCYWTEFT
|
7.9 | IC50 | 2 | — | |
DCDKXVMMAAIMRA
|
7.8 | IC50 | 3 | — | |
MGMOBQWMSWOTLL
|
7.8 | IC50 | 3 | — | |
BYKVUESQXQHBEP
|
7.8 | IC50 | 7 | — | |
FCJGMZMSVIAAJU
|
7.8 | IC50 | 9 | — | |
NBCDTZGTPATHKN
|
7.8 | IC50 | 2 | — | |
WWTRFWLRGARRAD
|
7.8 | IC50 | 10 | — | |
UIARLYUEJFELEN
|
7.8 | Kd | 289 | Yes | |
XSGDOSCYEQRDBE
|
7.8 | IC50 | 3 | — | |
DYNHJHQFHQTFTP
|
7.8 | Kd | 38 | — | |
GTSDNTZRPRBMTP
|
7.8 | IC50 | 3 | — | |
JPVJPXAQFGYJDI
|
7.8 | IC50 | 3 | — | |
JZTOUVBEZONDKA
|
7.8 | Ki | 80 | — | |
UKMGZRUGIXWOJQ
|
7.8 | IC50 | 3 | — | |
UNQLMLVHYGLKLZ
|
7.8 | IC50 | 2 | — | |
CNFUDCYXMQHQFO
|
7.8 | IC50 | 3 | — | |
YPGZOVPNRGMYIT
|
7.8 | IC50 | 3 | — | |
QQWUGDVOUVUTOY
|
7.8 | Kd | 231 | Yes | |
JKDJAOQUTMBBQB
|
7.8 | IC50 | 5 | — | |
UKXHMXAKNAXPBS
|
7.7 | IC50 | 3 | — | |
SVJBHQPXESBDEQ
|
7.7 | IC50 | 9 | — | |
CSZAJEXPQFERTK
|
7.7 | IC50 | 10 | — | |
JFGUWNUTXLHXTB
|
7.7 | IC50 | 2 | — |