Target Details
| UniProt AC | Q9H0K1 |
|---|---|
| Gene Symbol | SIK2 |
| Protein Name | Serine/threonine-protein kinase SIK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF23312 (UBA_SIK3) |
Summary
- Multi-target molecules 250
- Clinical molecules 23
- Avg pChEMBL 7.83
KEGG Pathways (1)
Active Molecules (250)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XVNZURGXHLXJIR
|
8.8 | IC50 | 3 | — | |
QBSNPDJXAMBWIZ
|
8.7 | IC50 | 3 | — | |
VCQQIZTUIHARTH
|
8.7 | IC50 | 3 | — | |
XOZORSAAPNHXFP
|
8.7 | IC50 | 3 | — | |
AQSSMEORRLJZLU
|
8.7 | Kd | 34 | Yes | |
AQXQPESYCSEOOG
|
8.7 | IC50 | 3 | — | |
GRPZYURNHYVZBO
|
8.7 | IC50 | 3 | — | |
HSYDEPQAUCZNGP
|
8.7 | IC50 | 3 | — | |
PNAUGSWMKOHDJF
|
8.7 | IC50 | 3 | — | |
OYDTWNVVTPPDDO
|
8.6 | IC50 | 3 | — | |
VNWAWEZKWMFEJY
|
8.6 | IC50 | 6 | — | |
UNBNKYSPLOMIOY
|
8.6 | IC50 | 7 | — | |
SVNQOEFGBNGPSZ
|
8.6 | IC50 | 3 | — | |
ZMAJVXKEVISHMQ
|
8.6 | IC50 | 9 | — | |
MMGVIQXQPXLHQK
|
8.6 | IC50 | 3 | — | |
RPDJXKWOAHHTBX
|
8.6 | IC50 | 3 | — | |
XCGUGTWHQADPNS
|
8.6 | IC50 | 3 | — | |
OMDTWHBLOYOZGL
|
8.5 | IC50 | 3 | — | |
MBBASLHNWYZIRZ
|
8.5 | IC50 | 3 | — | |
OSVUGUHRKMMBSE
|
8.5 | Kd | 170 | — | |
SIICZZZVCXGXGX
|
8.5 | IC50 | 3 | — | |
JVBRZBKYIRZVJE
|
8.5 | IC50 | 3 | — | |
ARXQRVVEKOEUEV
|
8.5 | IC50 | 3 | — | |
DNKJWTDFPIZFNK
|
8.5 | IC50 | 3 | — | |
XGEBOBAOVSOQCV
|
8.5 | IC50 | 10 | — | |
QYFGVVMJUHWKNB
|
8.5 | IC50 | 3 | — | |
UXTSNWGOMSEBTG
|
8.5 | IC50 | 2 | — | |
RGEJEFYGSBMYRS
|
8.4 | IC50 | 3 | — | |
QOOLIAIGEONMHK
|
8.4 | IC50 | 3 | — | |
SXMRTOWWEVQQSC
|
8.4 | IC50 | 3 | — | |
CAWABSRZIMATJO
|
8.4 | IC50 | 9 | — | |
UEQMHAFWQDRPMU
|
8.4 | IC50 | 3 | — | |
JLWGOAGEDWMEBT
|
8.4 | IC50 | 10 | — | |
JLWGOAGEDWMEBT
|
8.4 | IC50 | 10 | — | |
NXSJMRCTGYTSTK
|
8.4 | Kd | 200 | — | |
WRPKJPATUZRQFL
|
8.4 | IC50 | 3 | — | |
AQXQPESYCSEOOG
|
8.3 | IC50 | 3 | — | |
VFDIZCUBJRZYFL
|
8.3 | IC50 | 3 | — | |
KNOCCCXGASNIAF
|
8.3 | IC50 | 3 | — | |
XPJFDYHVVLGXHY
|
8.3 | IC50 | 3 | — | |
XELNNUJRQXCODY
|
8.3 | IC50 | 3 | — | |
BHFWGYATBPONNI
|
8.3 | IC50 | 3 | — | |
FWRPKNVNQNONLF
|
8.3 | IC50 | 2 | — | |
ZXYITDGKYOBFAO
|
8.3 | IC50 | 3 | — | |
UEOOSASFOHAWBP
|
8.2 | IC50 | 2 | — | |
IIRJOBJKMBEOMH
|
8.2 | IC50 | 3 | — | |
KZVDQIXBUFBWLM
|
8.2 | IC50 | 3 | — | |
MJSHVHLADKXCML
|
8.2 | IC50 | 11 | — | |
SHMKAHZOTDZUIN
|
8.2 | IC50 | 3 | — | |
IVKGWWZSELOWKX
|
8.2 | IC50 | 3 | — |