Target Details
| UniProt AC | Q9H0K1 |
|---|---|
| Gene Symbol | SIK2 |
| Protein Name | Serine/threonine-protein kinase SIK2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF23312 (UBA_SIK3) |
Summary
- Multi-target molecules 250
- Clinical molecules 23
- Avg pChEMBL 7.83
KEGG Pathways (1)
Active Molecules (250)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QVUYJTWSZWCKHP
|
10.0 | IC50 | 3 | — | |
KDPXVKRYHKSBPY
|
9.7 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
9.4 | IC50 | 408 | — | |
AWLHPMOLJAWKDL
|
9.4 | IC50 | 3 | — | |
DYMFNPBLDKXKJA
|
9.4 | IC50 | 3 | — | |
VOYZWDQJVPQGCO
|
9.4 | IC50 | 9 | — | |
XHPICGSLCSAZKX
|
9.4 | IC50 | 3 | — | |
LTQKUGJNXFIXKC
|
9.4 | IC50 | 3 | — | |
HOKRUYIIDRQYFK
|
9.3 | IC50 | 3 | — | |
YOWQNRVRQMOXAT
|
9.3 | IC50 | 3 | — | |
YCOQHBLWDSAZRB
|
9.2 | IC50 | 3 | — | |
RZXPVLRGCBTJSU
|
9.2 | IC50 | 3 | — | |
HSQLWSUNRMTGGO
|
9.2 | IC50 | 3 | — | |
WXCYMIOQVROELY
|
9.2 | IC50 | 3 | — | |
NQANXDMJOUTFBB
|
9.2 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
9.2 | Ki | 118 | — | |
AZCVMDQKOWCQAG
|
9.2 | IC50 | 3 | — | |
WCLYSPWUHSZWOR
|
9.2 | IC50 | 3 | — | |
LYSXGFLZKDKZDF
|
9.2 | IC50 | 3 | — | |
PFTXFNSHFZLJNT
|
9.2 | IC50 | 17 | — | |
YATIMLFNGFQTCA
|
9.2 | IC50 | 3 | — | |
FGLQSISJARINNB
|
9.1 | IC50 | 3 | — | |
WMCHGBLGKMZDJD
|
9.1 | IC50 | 3 | — | |
RXHXLESLBWUVQS
|
9.1 | IC50 | 3 | — | |
NDNNIKHUOLIORS
|
9.1 | IC50 | 3 | — | |
WDNAXOPVZIEECR
|
9.1 | IC50 | 11 | — | |
JWADUJSXPDSTOX
|
9.0 | IC50 | 3 | — | |
AWVUPXUQWGNTHF
|
9.0 | IC50 | 3 | — | |
BIYKGGOFJOFQIZ
|
9.0 | IC50 | 3 | — | |
INXQKXZSUNICKV
|
9.0 | IC50 | 3 | — | |
OWRXHGAFWZFFCW
|
9.0 | Ki | 113 | — | |
WEHOIIGXTMKVRG
|
9.0 | IC50 | 3 | — | |
XUOIDCGCIMNQCG
|
9.0 | IC50 | 3 | — | |
YMSJZKSIBUPNHN
|
9.0 | IC50 | 3 | — | |
AEYQVJYAPMGHSF
|
9.0 | IC50 | 3 | — | |
BIYKGGOFJOFQIZ
|
9.0 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
9.0 | Kd | 213 | — | |
PZFORNOVSGDEAS
|
9.0 | IC50 | 3 | — | |
KAUKMJZXRPFGAB
|
8.9 | IC50 | 3 | — | |
OKSHQZCQVDERIF
|
8.9 | IC50 | 3 | — | |
FQZGWTSGSBKLBT
|
8.9 | IC50 | 3 | — | |
DEJPFOVGKKDPLD
|
8.8 | IC50 | 3 | — | |
OLULSQINUASNMI
|
8.8 | IC50 | 3 | — | |
BQKJBKRZMBOHNT
|
8.8 | IC50 | 3 | — | |
VATIVDMNNPRBCN
|
8.8 | IC50 | 3 | — | |
WKZOFECSVXLTOB
|
8.8 | IC50 | 3 | — | |
CAJPKOHOPAWXRV
|
8.8 | IC50 | 3 | — | |
FPNPNYBQZUNHGQ
|
8.8 | IC50 | 3 | — | |
CFNFPVIKPAPVOV
|
8.8 | IC50 | 3 | — | |
MXNBWDNCIZQCIL
|
8.8 | IC50 | 3 | — |