Target Details
| UniProt AC | Q9H0J9 |
|---|---|
| Gene Symbol | PARP12 |
| Protein Name | Protein mono-ADP-ribosyltransferase PARP12 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00644 (PARP) PF24356 (WHD_PARP12) PF02825 (WWE) PF23466 (WWE_4) PF25261 (zf-CCCH_PARP12) |
Summary
- Multi-target molecules 10
- Clinical molecules 0
- Avg pChEMBL 6.75
Active Molecules (10)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
STSCRAGBCYODMY
|
7.8 | IC50 | 8 | — | |
UQZCQKXJAXKZQH
|
7.6 | IC50 | 4 | — | |
PCHKPVIQAHNQLW
|
7.1 | IC50 | 8 | — | |
FSNNMBVVDWKKCB
|
6.8 | IC50 | 6 | — | |
UYJZZVDLGDDTCL
|
6.6 | IC50 | 8 | — | |
BANSZVBMEHYKAV
|
6.4 | IC50 | 4 | — | |
JLVRTMBMCWYGAL
|
6.4 | IC50 | 7 | — | |
BMPSOKZAIFFMLK
|
6.3 | IC50 | 6 | — | |
ZXYKQNYSXHNQMV
|
6.2 | IC50 | 6 | — | |
FDLYAMZZIXQODN
|
6.2 | IC50 | 11 | — |