Target Details
| UniProt AC | Q9H093 |
|---|---|
| Gene Symbol | NUAK2 |
| Protein Name | NUAK family SNF1-like kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 42
- Clinical molecules 14
- Avg pChEMBL 7.18
Associated Diseases (1)
Active Molecules (42)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
10.1 | Kd | 213 | — | |
YPJRHEKCFKOVRT
|
9.2 | Kd | 12 | — | |
UIARLYUEJFELEN
|
9.0 | Kd | 289 | Yes | |
QQWUGDVOUVUTOY
|
8.9 | Kd | 231 | Yes | |
HKSZLNNOFSGOKW
|
8.8 | IC50 | 408 | — | |
RSFALMGMTQBFJZ
|
8.5 | Kd | 9 | — | |
ITTRLTNMFYIYPA
|
8.0 | Kd | 17 | — | |
NXSJMRCTGYTSTK
|
8.0 | Kd | 200 | — | |
OSVUGUHRKMMBSE
|
8.0 | Kd | 170 | — | |
XZXHXSATPCNXJR
|
7.7 | Kd | 165 | Yes | |
ZHJGWYRLJUCMRT
|
7.6 | Kd | 18 | — | |
RYYNGWLOYLRZLK
|
7.6 | Kd | 45 | — | |
XKFTZKGMDDZMJI
|
7.6 | Kd | 64 | Yes | |
KDKUVYLMPJIGKA
|
7.6 | Kd | 91 | Yes | |
JOOXLOJCABQBSG
|
7.3 | Kd | 139 | — | |
YYLKKYCXAOBSRM
|
7.3 | Kd | 191 | — | |
BMGQWWVMWDBQGC
|
7.2 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
7.2 | Kd | 91 | Yes | |
NHHQJBCNYHBUSI
|
7.2 | Kd | 220 | — | |
KGPGFQWBCSZGEL
|
7.1 | Kd | 59 | Yes | |
SDGJBAUIGHSMRI
|
7.0 | IC50 | 3 | — | |
KTEIFNKAUNYNJU
|
6.9 | Kd | 114 | — | |
LZUYOYKXEXENTQ
|
6.9 | IC50 | 5 | — | |
GUBJNPWVIUFSTR
|
6.9 | Kd | 103 | — | |
PIQCTGMSNWUMAF
|
6.9 | Kd | 137 | Yes | |
JWNPDZNEKVCWMY
|
6.8 | Kd | 57 | Yes | |
WINHZLLDWRZWRT
|
6.8 | Kd | 201 | Yes | |
UBPYILGKFZZVDX
|
6.7 | Kd | 130 | Yes | |
HFNKQEVNSGCOJV
|
6.5 | Kd | 65 | — | |
ZCBUQCWBWNUWSU
|
6.5 | Kd | 59 | — | |
CTNPALGJUAXMMC
|
6.4 | Kd | 151 | — | |
UJLAWZDWDVHWOW
|
6.4 | Kd | 16 | — | |
ZZSBPGIGIUFJRA
|
6.4 | Kd | 46 | — | |
FWLMVFUGMHIOAA
|
6.3 | Kd | 26 | — | |
GCIKSSRWRFVXBI
|
6.3 | Kd | 109 | Yes | |
WKDACQVEJIVHMZ
|
6.2 | Kd | 46 | — | |
OEZHSZIDGUKBRK
|
6.0 | IC50 | 10 | — | |
OYONTEXKYJZFHA
|
6.0 | Kd | 69 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
ZCCPLJOKGAACRT
|
6.0 | Kd | 599 | — |