Target Details
| UniProt AC | Q9GUA8 |
|---|---|
| Gene Symbol | HD1 |
| Protein Name | Histone deacetylase |
| Organism | Cryptosporidium parvum |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00850 (Hist_deacetyl) |
Summary
- Multi-target molecules 25
- Clinical molecules 13
- Avg pChEMBL 8.07
Active Molecules (25)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UCPPLLAVVTUHRE
|
9.7 | IC50 | 14 | Yes | |
JPJYOPNEGMWFJL
|
9.1 | IC50 | 15 | Yes | |
MGSMSINQVPOBFG
|
9.1 | IC50 | 12 | — | |
BHYPIIUJEQHYIP
|
9.0 | IC50 | 14 | Yes | |
JWOGUUIOCYMBPV
|
9.0 | IC50 | 17 | Yes | |
JMMPUTVKLCAIID
|
8.7 | IC50 | 15 | Yes | |
HWYVSKGWENBBBO
|
8.5 | IC50 | 14 | Yes | |
BCSAECULXJTTAB
|
8.4 | IC50 | 12 | — | |
GIVUNOYVRYOCFE
|
8.4 | IC50 | 13 | Yes | |
HVAMCPMMTPHGBZ
|
8.4 | IC50 | 12 | — | |
IEVZGTIIJVLPRE
|
8.4 | IC50 | 15 | Yes | |
IDNMSLGHIWCDPW
|
8.3 | IC50 | 2 | — | |
RZIVQAPDZCRFHM
|
8.3 | IC50 | 2 | — | |
OHZAUIQSIDAXOV
|
8.0 | IC50 | 2 | — | |
QIRFIQOIPIMCJZ
|
8.0 | IC50 | 15 | Yes | |
ONHTZJLXGIZPCI
|
7.7 | IC50 | 15 | Yes | |
QYPHTJRLIJBSGN
|
7.6 | IC50 | 2 | — | |
VXHZOOMBKKPXQS
|
7.5 | IC50 | 12 | — | |
CSQVBMSEOLWQFW
|
7.5 | IC50 | 13 | Yes | |
MUZSIPXZOGAVSZ
|
7.3 | IC50 | 15 | Yes | |
LPLNOQJRDCBMJX
|
7.3 | IC50 | 15 | Yes | |
SOGXSPMNYVWNRR
|
7.0 | IC50 | 2 | — | |
SUWIMJYUHRRXMN
|
7.0 | IC50 | 2 | — | |
VDYRVGYMGXRGMO
|
6.8 | IC50 | 2 | — | |
WSPZAXPNRNZYQV
|
6.7 | IC50 | 2 | — |