Target Details
| UniProt AC | Q9F663 |
|---|---|
| Gene Symbol | KPC-2 |
| Protein Name | Carbapenem-hydrolyzing beta-lactamase KPC-2 |
| Organism | Klebsiella pneumoniae |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF13354 (Beta-lactamase2) |
Summary
- Multi-target molecules 3
- Clinical molecules 0
- Avg pChEMBL 6.41
Top Co-occurrence Targets
- blaCTX-M-14 2 shared
- blaTEM-1 2 shared
- OXA-1 2 shared
- ampC 2 shared
- blaUOE-1 1 shared
- bla OXY 1 shared
- blaTEM-1 1 shared
- blaTEM-125 1 shared
- 1 shared
- imiA 1 shared
Active Molecules (3)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NDCUAPJVLWFHHB
|
6.7 | IC50 | 8 | — | |
LPQZKKCYTLCDGQ
|
6.4 | IC50 | 15 | — | |
RSBPYSTVZQAADE
|
6.1 | IC50 | 4 | — |