Target Details
| UniProt AC | Q9EXV5 |
|---|---|
| Gene Symbol | blaUOE-1 |
| Protein Name | Beta-lactamase |
| Organism | Escherichia coli |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF13354 (Beta-lactamase2) |
Summary
- Multi-target molecules 2
- Clinical molecules 0
- Avg pChEMBL 8.38
Top Co-occurrence Targets
- bla OXY 2 shared
- blaCTX-M-53 2 shared
- OXA-1 2 shared
- blaZ 2 shared
- blaGES-13 2 shared
- blaSCO-1 2 shared
- KPC-2 1 shared
- blaTEM-1 1 shared
- blaTEM-125 1 shared
- 1 shared
Active Molecules (2)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LPQZKKCYTLCDGQ
|
8.7 | IC50 | 15 | — | |
HZZVJAQRINQKSD
|
8.1 | IC50 | 13 | — |