Target Details
| UniProt AC | Q9C098 |
|---|---|
| Gene Symbol | DCLK3 |
| Protein Name | Serine/threonine-protein kinase DCLK3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 20
- Clinical molecules 6
- Avg pChEMBL 6.83
Active Molecules (20)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UJLAWZDWDVHWOW
|
8.3 | Kd | 16 | — | |
JOOXLOJCABQBSG
|
7.9 | Kd | 139 | — | |
QQWUGDVOUVUTOY
|
7.8 | Kd | 231 | Yes | |
HKSZLNNOFSGOKW
|
7.8 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
7.8 | Kd | 213 | — | |
NXSJMRCTGYTSTK
|
7.2 | Kd | 200 | — | |
YYLKKYCXAOBSRM
|
7.1 | Kd | 191 | — | |
OSVUGUHRKMMBSE
|
7.0 | Kd | 170 | — | |
KGPGFQWBCSZGEL
|
7.0 | Kd | 59 | Yes | |
WINHZLLDWRZWRT
|
7.0 | Kd | 201 | Yes | |
CTNPALGJUAXMMC
|
6.6 | Kd | 151 | — | |
HFNKQEVNSGCOJV
|
6.6 | Kd | 65 | — | |
NHHQJBCNYHBUSI
|
6.2 | Kd | 220 | — | |
JRNJNYBQQYBCLE
|
6.2 | Kd | 40 | Yes | |
XZXHXSATPCNXJR
|
6.1 | Kd | 165 | Yes | |
MFAQYJIYDMLAIM
|
6.1 | Kd | 130 | Yes | |
ITTRLTNMFYIYPA
|
6.0 | Kd | 17 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |