Target Details
| UniProt AC | Q9BZL6 |
|---|---|
| Gene Symbol | PRKD2 |
| Protein Name | Serine/threonine-protein kinase D2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00169 (PH) PF00069 (Pkinase) PF25525 (Ubiquitin_PRKD1_N) |
Summary
- Multi-target molecules 219
- Clinical molecules 14
- Avg pChEMBL 6.87
KEGG Pathways (3)
Active Molecules (219)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JZSWBZHJDCDLHK
|
6.3 | Ki | 10 | — | |
OADRBDVURCEKRP
|
6.3 | Ki | 44 | — | |
OWDRQHVEJIYVOI
|
6.3 | Ki | 47 | — | |
QAJPIJHWTGPUNZ
|
6.3 | Ki | 37 | — | |
VNGYQBMDQMDALH
|
6.3 | Ki | 25 | — | |
WPHKIQPVPYJNAX
|
6.3 | Ki | 81 | — | |
WZZXMNBOPNKKSX
|
6.3 | Ki | 10 | — | |
XBAIEEJJCJHBDL
|
6.3 | Ki | 17 | — | |
XPHWIERLJBFPFV
|
6.3 | Ki | 69 | — | |
XSRHBCYNCKAFKS
|
6.3 | Ki | 45 | — | |
YMSZHISTTIUBDG
|
6.3 | Ki | 7 | — | |
XQVVPGYIWAGRNI
|
6.3 | Kd | 34 | — | |
WXGCJNLWHYWDFU
|
6.3 | IC50 | 3 | — | |
JTVBXQAYBIJXRP
|
6.2 | Kd | 20 | — | |
XQJWTJLJEYIUDZ
|
6.2 | IC50 | 2 | — | |
AOBLBPWPSKBHSI
|
6.2 | Ki | 55 | — | |
CFBADDSSFSYJPF
|
6.2 | Ki | 23 | — | |
CXBBWVXSZINRCS
|
6.2 | Ki | 41 | — | |
DKXHSOUZPMHNIZ
|
6.2 | Ki | 51 | Yes | |
FGWOKLCRQJXPPQ
|
6.2 | Ki | 14 | — | |
IPKHSYHXXAIZDD
|
6.2 | Ki | 18 | — | |
NHHQJBCNYHBUSI
|
6.2 | Ki | 220 | — | |
RKKIDHHGKNGTQI
|
6.2 | Ki | 28 | — | |
UCOWZARZLHNDKP
|
6.2 | Ki | 8 | — | |
UEIRKXUBXCSHJE
|
6.2 | Ki | 19 | — | |
USHMNZBDAOGLMB
|
6.2 | Ki | 26 | — | |
UUWNXFJBBYAMDT
|
6.2 | Ki | 46 | — | |
XIOOJUQFJYPVLA
|
6.2 | Ki | 17 | — | |
XJSFDMGICAWQFS
|
6.2 | Ki | 60 | — | |
ZKHDDJKHTPLPOQ
|
6.2 | Ki | 62 | — | |
ZVWRFVCNQOECJS
|
6.2 | Ki | 71 | — | |
ZYTFPHRVOZXPGZ
|
6.2 | Ki | 30 | — | |
XZXHXSATPCNXJR
|
6.1 | Kd | 165 | Yes | |
WLYQNZYLNRAMFN
|
6.1 | IC50 | 2 | — | |
FQYLJBVSYHZWLT
|
6.1 | Ki | 35 | Yes | |
FTIAKTLRFKSDFR
|
6.1 | Ki | 10 | Yes | |
GDQXJQSQYMMKRA
|
6.1 | IC50 | 15 | — | |
ICDHVAJOGIGIOI
|
6.1 | Ki | 5 | — | |
IJNGXROUMFEKDB
|
6.1 | Ki | 39 | — | |
KNACLJBHKVSTDL
|
6.1 | Ki | 40 | — | |
SHENEEFOURUIBP
|
6.1 | Ki | 29 | — | |
WIHAOLDOGQOGIU
|
6.1 | Ki | 5 | — | |
XHORJSJFHVABEA
|
6.1 | Ki | 49 | — | |
ZCBUQCWBWNUWSU
|
6.0 | Kd | 59 | — | |
HFTWWDARPWZARK
|
6.0 | IC50 | 3 | — | |
RYYNGWLOYLRZLK
|
6.0 | Kd | 45 | — | |
CSDDCHPGQGWRLI
|
6.0 | Ki | 5 | Yes | |
JPOSFPUHBHRUAX
|
6.0 | IC50 | 40 | Yes | |
ODPGGGTTYSGTGO
|
6.0 | Kd | 153 | — | |
DPRGOXVMSNDADU
|
6.0 | Ki | 16 | — |