Target Details
| UniProt AC | Q9BZL6 |
|---|---|
| Gene Symbol | PRKD2 |
| Protein Name | Serine/threonine-protein kinase D2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00169 (PH) PF00069 (Pkinase) PF25525 (Ubiquitin_PRKD1_N) |
Summary
- Multi-target molecules 219
- Clinical molecules 14
- Avg pChEMBL 6.87
KEGG Pathways (3)
Active Molecules (219)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VXYDJXMHISGSDA
|
6.8 | Ki | 59 | — | |
FWXIKQAZCDAIKV
|
6.8 | IC50 | 3 | — | |
WMFOYAZROOMVDL
|
6.8 | IC50 | 3 | — | |
NDIUYMHNCUTVGE
|
6.8 | Ki | 25 | — | |
FKJNUFATJIQZEN
|
6.7 | IC50 | 2 | — | |
XLSYZSRXVVCHLS
|
6.7 | Kd | 48 | — | |
CLEGDJQQHUTCOW
|
6.7 | Ki | 43 | — | |
JRZRHWNUPAZFMZ
|
6.7 | IC50 | 2 | — | |
MIKAKZKNMYZLDX
|
6.7 | Ki | 42 | — | |
WVFWTUJEHMVUBG
|
6.7 | Ki | 25 | — | |
XNEPVLVYFUGJLF
|
6.7 | Ki | 27 | — | |
YEHCNYAQEBQCCS
|
6.7 | Ki | 74 | — | |
PNZJIQBIMCZAKU
|
6.7 | IC50 | 3 | — | |
LQERXZYSNKIMFN
|
6.7 | IC50 | 2 | — | |
NVHXHWFKRHCFCI
|
6.6 | IC50 | 3 | — | |
KWKHZFAYBPSEGP
|
6.6 | IC50 | 2 | — | |
LOLPPWBBNUVNQZ
|
6.6 | Kd | 97 | Yes | |
DFMCXVONDDGQIY
|
6.6 | Ki | 66 | — | |
GQLWKGVBOIYMTN
|
6.6 | Ki | 35 | — | |
UMTWTCVTRDYHQQ
|
6.6 | Ki | 56 | — | |
WDXXELAFEZBSNE
|
6.6 | IC50 | 2 | — | |
XFWUTMHVDGPWLH
|
6.6 | Ki | 75 | — | |
XJJYJNMNYDNXNO
|
6.6 | Ki | 23 | — | |
LSUPQYXXQGNJGE
|
6.6 | IC50 | 2 | — | |
XKVKEBRJQBYODL
|
6.6 | IC50 | 2 | — | |
AACFPJSJOWQNBN
|
6.5 | IC50 | 4 | — | |
HZCVZGCAUBUBST
|
6.5 | IC50 | 3 | — | |
AILRADAXUVEEIR
|
6.5 | IC50 | 75 | — | |
BPNUQXPIQBZCMR
|
6.5 | Ki | 60 | — | |
GUBJNPWVIUFSTR
|
6.5 | Kd | 103 | — | |
GWJHMRBQEUHFOC
|
6.5 | Ki | 42 | — | |
KOHNRDPXFDZZJF
|
6.5 | Ki | 31 | — | |
NKGLJTITEFZKAN
|
6.5 | Ki | 35 | — | |
ORUUEFDGYYTXAF
|
6.5 | Ki | 26 | — | |
OUJZYQBEFNDJQN
|
6.5 | Ki | 71 | — | |
RKUKAACYUCUJEE
|
6.5 | Ki | 58 | — | |
XQVVPGYIWAGRNI
|
6.5 | Ki | 19 | — | |
XYZNKCSDQRKAFR
|
6.5 | Ki | 53 | — | |
ZCCPLJOKGAACRT
|
6.5 | Kd | 599 | — | |
LLEOOSLUHRQCHZ
|
6.5 | IC50 | 6 | — | |
WINHZLLDWRZWRT
|
6.4 | Kd | 201 | Yes | |
CXZZKTFGTNQHGD
|
6.4 | Ki | 4 | — | |
GHPFQRTVUDXWCC
|
6.4 | Ki | 35 | — | |
UAQJVFADAYIBGC
|
6.4 | Ki | 23 | — | |
UDFDIIVNIYWXDM
|
6.4 | Ki | 74 | — | |
WINHZLLDWRZWRT
|
6.4 | Ki | 66 | — | |
LTWPQYSXDJCNBR
|
6.4 | IC50 | 3 | — | |
GGFLGGNNYKCRAV
|
6.3 | IC50 | 3 | — | |
VXBAJLGYBMTJCY
|
6.3 | Kd | 34 | Yes | |
FLEAYYMORDPWAJ
|
6.3 | Ki | 90 | — |