Target Details
| UniProt AC | Q9BZL6 |
|---|---|
| Gene Symbol | PRKD2 |
| Protein Name | Serine/threonine-protein kinase D2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00169 (PH) PF00069 (Pkinase) PF25525 (Ubiquitin_PRKD1_N) |
Summary
- Multi-target molecules 219
- Clinical molecules 14
- Avg pChEMBL 6.87
KEGG Pathways (3)
Active Molecules (219)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AWJAAKKEYXUCFY
|
7.3 | IC50 | 5 | — | |
LSEXYAQECWMUPY
|
7.3 | IC50 | 3 | — | |
AKWVKIGCMCHYJT
|
7.3 | Ki | 8 | — | |
FTCSRLCKGZJDCK
|
7.3 | IC50 | 3 | — | |
GCBJDOWIQHMCMR
|
7.3 | Ki | 84 | — | |
GCYXEGSPUDSZJY
|
7.3 | Ki | 82 | — | |
LRZYYIZFBXFSJB
|
7.3 | Ki | 69 | — | |
YEOMJKKERMIQSA
|
7.3 | IC50 | 2 | — | |
WHROQBPMBHWWTB
|
7.3 | IC50 | 3 | — | |
XDJCLCLBSGGNKS
|
7.2 | Kd | 21 | — | |
DHUAGGSHTKPOHU
|
7.2 | IC50 | 3 | — | |
LRYNHRWGDADZKP
|
7.2 | IC50 | 3 | — | |
SFSGIDJMRRLJFG
|
7.2 | IC50 | 3 | — | |
ZIATUPKJNZVSLT
|
7.2 | IC50 | 3 | — | |
RYYNGWLOYLRZLK
|
7.2 | Ki | 104 | — | |
ZVKJUDYDWABBFR
|
7.2 | IC50 | 3 | — | |
DKZYXHCYPUVGAF
|
7.2 | Kd | 112 | — | |
HKSZLNNOFSGOKW
|
7.1 | Kd | 213 | — | |
VAVGLCQDZFLPHS
|
7.1 | IC50 | 3 | — | |
CLRFYTGANQZOBS
|
7.1 | Ki | 41 | — | |
FDVSOQRNTAPCHB
|
7.1 | Ki | 40 | — | |
MGNQNQOSSLCUFP
|
7.1 | Ki | 12 | — | |
MVJMMLFMPWITEJ
|
7.1 | Ki | 110 | — | |
NXSJMRCTGYTSTK
|
7.1 | Kd | 200 | — | |
PCQMERRARZKTPW
|
7.1 | Ki | 68 | — | |
SFSGIDJMRRLJFG
|
7.1 | IC50 | 3 | — | |
BERLXWPRSBJFHO
|
7.0 | IC50 | 4 | — | |
RBZLXANOQRQGTN
|
7.0 | IC50 | 3 | — | |
CNLCKMDXRXVYMV
|
7.0 | IC50 | 3 | — | |
OWRXHGAFWZFFCW
|
7.0 | Ki | 113 | — | |
ZUYALLZMSFUHFE
|
7.0 | IC50 | 3 | — | |
HUXYBQXJVXOMKX
|
7.0 | Kd | 28 | — | |
YZAJDKHTPRXEKJ
|
7.0 | IC50 | 2 | — | |
BRBMDFAROPPCNO
|
6.9 | IC50 | 2 | — | |
CKVWQORGCCEYHS
|
6.9 | Ki | 50 | — | |
HHSVICUMCOBRPT
|
6.9 | Ki | 33 | — | |
JWQOJVOKBAAAAR
|
6.9 | Ki | 29 | — | |
JZTOUVBEZONDKA
|
6.9 | Ki | 80 | — | |
LYNBNVBMAGDJRW
|
6.9 | Ki | 81 | — | |
WYOMXSAYYXBPMN
|
6.9 | Ki | 24 | — | |
VJHWVSYYFZRUEK
|
6.9 | IC50 | 3 | — | |
XSHQBIXMLULFEV
|
6.9 | IC50 | 13 | — | |
ZHMXXVNQAFCXKK
|
6.9 | IC50 | 15 | — | |
CSGQVNMSRKWUSH
|
6.8 | Kd | 21 | — | |
KGMSYXGSYGEHIS
|
6.8 | IC50 | 4 | — | |
OSVUGUHRKMMBSE
|
6.8 | Kd | 170 | — | |
XKVKEBRJQBYODL
|
6.8 | IC50 | 2 | — | |
FOLSZCLZVLICGG
|
6.8 | IC50 | 2 | — | |
KRIUNPBAQZGFQA
|
6.8 | Ki | 76 | — | |
QQWUGDVOUVUTOY
|
6.8 | Kd | 231 | Yes |