Target Details
UniProt ACQ9BZL6
Gene SymbolPRKD2
Protein NameSerine/threonine-protein kinase D2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00130 (C1_1) PF00169 (PH) PF00069 (Pkinase) PF25525 (Ubiquitin_PRKD1_N)
Summary
  • Multi-target molecules 219
  • Clinical molecules 14
  • Avg pChEMBL 6.87
Top Co-occurrence Targets
Active Molecules (219)
InChIKey pChEMBL Type Targets Clinical
IHAKCSKGCPKKPZ 9.0 IC50 2
MTXHXAFTVABHOY 9.0 IC50 3
XVKPIWUWUZOHIR 8.7 IC50 3
DIZACSOTRSXCHC 8.7 IC50 4
VWVQWSIGDZWPIL 8.7 IC50 2
XBDRAUPLGHAFCU 8.7 IC50 3
ZYRFDYUCAPSAAJ 8.7 IC50 2
HKSZLNNOFSGOKW 8.6 Ki 118
SCJXQZZYGYLKJG 8.6 IC50 3
AQSSMEORRLJZLU 8.5 Kd 34 Yes
QQXZJQAEELFYDV 8.3 IC50 2
RQVKVJIRFKVPBF 8.2 Ki 13
BRBMDFAROPPCNO 8.2 IC50 2
PIPGGBLVUJYMED 8.2 IC50 3
HCMOZLPTNMKKAS 8.2 IC50 3
KKMZQQWZVBKDFC 8.1 IC50 3
QHBRARNRIAKCGO 8.1 IC50 2
RJZDECGDCKOHBV 8.1 Ki 70
UQFRSHRWRKYNDE 8.1 Ki 17 Yes
VDRJYOAEHZMFEB 8.1 IC50 3
UIARLYUEJFELEN 8.1 Kd 289 Yes
NCAVLXJPDIQUIS 8.1 IC50 3
SCJXQZZYGYLKJG 8.1 IC50 3
XNWDRALEEPGBHB 8.1 IC50 3
YKWMQNUCOUUHQO 8.1 IC50 3
HKSZLNNOFSGOKW 8.0 IC50 408
MZIOLOXGGOLJMJ 7.9 Ki 12
NLUPJKQOKWBWFC 7.9 Ki 69
BSFNGHCTZDCQBF 7.8 Ki 93
VWVYILCFSYNJHF 7.8 Ki 49
ZACCEWDQLIBKAZ 7.8 IC50 2
MESYXTDMWTWQNS 7.8 IC50 2
WXGCJNLWHYWDFU 7.8 IC50 3
FUMCKNCUEAQHCV 7.7 Ki 103
VLEFVPMCVJDTHZ 7.7 Ki 13
ADMFLILDQJSEIK 7.6 Ki 72
HMBDNAGIIDHKKM 7.6 Ki 9
AYCPARAPKDAOEN 7.6 IC50 73
KOZFSFOOLUUIGY 7.5 Kd 88 Yes
MWKSRKSEWLRPBL 7.5 Kd 1075
VBWZGQKYVCFADL 7.5 IC50 3
CHTMRWQLNNRRFJ 7.5 Ki 70
YWTBGJGMTBHQTM 7.5 Ki 65
BFSMGDJOXZAERB 7.5 Kd 33
GTWNYADDKACXSW 7.5 IC50 3
HXYGELZVZAPWID 7.5 IC50 3
NJPWCTYVEJIQBM 7.4 Ki 72
OWFLADWRSCINST 7.4 Ki 30
YMIJUBCSOKSFRU 7.4 Ki 87
CEWOYNHYISZPFC 7.4 IC50 3
2D structure