Target Details
| UniProt AC | Q9BZL6 |
|---|---|
| Gene Symbol | PRKD2 |
| Protein Name | Serine/threonine-protein kinase D2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00130 (C1_1) PF00169 (PH) PF00069 (Pkinase) PF25525 (Ubiquitin_PRKD1_N) |
Summary
- Multi-target molecules 219
- Clinical molecules 14
- Avg pChEMBL 6.87
KEGG Pathways (3)
Active Molecules (219)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IHAKCSKGCPKKPZ
|
9.0 | IC50 | 2 | — | |
MTXHXAFTVABHOY
|
9.0 | IC50 | 3 | — | |
XVKPIWUWUZOHIR
|
8.7 | IC50 | 3 | — | |
DIZACSOTRSXCHC
|
8.7 | IC50 | 4 | — | |
VWVQWSIGDZWPIL
|
8.7 | IC50 | 2 | — | |
XBDRAUPLGHAFCU
|
8.7 | IC50 | 3 | — | |
ZYRFDYUCAPSAAJ
|
8.7 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
8.6 | Ki | 118 | — | |
SCJXQZZYGYLKJG
|
8.6 | IC50 | 3 | — | |
AQSSMEORRLJZLU
|
8.5 | Kd | 34 | Yes | |
QQXZJQAEELFYDV
|
8.3 | IC50 | 2 | — | |
RQVKVJIRFKVPBF
|
8.2 | Ki | 13 | — | |
BRBMDFAROPPCNO
|
8.2 | IC50 | 2 | — | |
PIPGGBLVUJYMED
|
8.2 | IC50 | 3 | — | |
HCMOZLPTNMKKAS
|
8.2 | IC50 | 3 | — | |
KKMZQQWZVBKDFC
|
8.1 | IC50 | 3 | — | |
QHBRARNRIAKCGO
|
8.1 | IC50 | 2 | — | |
RJZDECGDCKOHBV
|
8.1 | Ki | 70 | — | |
UQFRSHRWRKYNDE
|
8.1 | Ki | 17 | Yes | |
VDRJYOAEHZMFEB
|
8.1 | IC50 | 3 | — | |
UIARLYUEJFELEN
|
8.1 | Kd | 289 | Yes | |
NCAVLXJPDIQUIS
|
8.1 | IC50 | 3 | — | |
SCJXQZZYGYLKJG
|
8.1 | IC50 | 3 | — | |
XNWDRALEEPGBHB
|
8.1 | IC50 | 3 | — | |
YKWMQNUCOUUHQO
|
8.1 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
8.0 | IC50 | 408 | — | |
MZIOLOXGGOLJMJ
|
7.9 | Ki | 12 | — | |
NLUPJKQOKWBWFC
|
7.9 | Ki | 69 | — | |
BSFNGHCTZDCQBF
|
7.8 | Ki | 93 | — | |
VWVYILCFSYNJHF
|
7.8 | Ki | 49 | — | |
ZACCEWDQLIBKAZ
|
7.8 | IC50 | 2 | — | |
MESYXTDMWTWQNS
|
7.8 | IC50 | 2 | — | |
WXGCJNLWHYWDFU
|
7.8 | IC50 | 3 | — | |
FUMCKNCUEAQHCV
|
7.7 | Ki | 103 | — | |
VLEFVPMCVJDTHZ
|
7.7 | Ki | 13 | — | |
ADMFLILDQJSEIK
|
7.6 | Ki | 72 | — | |
HMBDNAGIIDHKKM
|
7.6 | Ki | 9 | — | |
AYCPARAPKDAOEN
|
7.6 | IC50 | 73 | — | |
KOZFSFOOLUUIGY
|
7.5 | Kd | 88 | Yes | |
MWKSRKSEWLRPBL
|
7.5 | Kd | 1075 | — | |
VBWZGQKYVCFADL
|
7.5 | IC50 | 3 | — | |
CHTMRWQLNNRRFJ
|
7.5 | Ki | 70 | — | |
YWTBGJGMTBHQTM
|
7.5 | Ki | 65 | — | |
BFSMGDJOXZAERB
|
7.5 | Kd | 33 | — | |
GTWNYADDKACXSW
|
7.5 | IC50 | 3 | — | |
HXYGELZVZAPWID
|
7.5 | IC50 | 3 | — | |
NJPWCTYVEJIQBM
|
7.4 | Ki | 72 | — | |
OWFLADWRSCINST
|
7.4 | Ki | 30 | — | |
YMIJUBCSOKSFRU
|
7.4 | Ki | 87 | — | |
CEWOYNHYISZPFC
|
7.4 | IC50 | 3 | — |