Target Details
| UniProt AC | Q9BZ95 |
|---|---|
| Gene Symbol | NSD3 |
| Protein Name | Histone-lysine N-methyltransferase NSD3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17907 (AWS) PF17982 (C5HCH) PF23011 (PHD-1st_NSD) PF22908 (PHD_NSD) PF23004 (PHDvar_NSD) PF00855 (PWWP) PF00856 (SET) |
Summary
- Multi-target molecules 12
- Clinical molecules 0
- Avg pChEMBL 8.14
KEGG Pathways (2)
Active Molecules (12)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DGGOQICQTAGRMC
|
9.0 | IC50 | 3 | — | |
FUEGZWGKKBGDBO
|
9.0 | IC50 | 3 | — | |
NKBVGYWANONFTE
|
9.0 | IC50 | 2 | — | |
OPJPZRUHVUFNAY
|
9.0 | IC50 | 3 | — | |
PIFXSVGCYBHXHR
|
9.0 | IC50 | 2 | — | |
RITHSQHPTNJAHO
|
9.0 | IC50 | 2 | — | |
WLGCCCLQJAMXCP
|
9.0 | IC50 | 3 | — | |
JXTDBIVBSAFNBJ
|
7.3 | Kd | 2 | — | |
AAAQFGUYHFJNHI
|
7.3 | IC50 | 252 | — | |
WYAGGMZTARRIDX
|
7.0 | Kd | 2 | — | |
YELBNEVEPNGEGQ
|
7.0 | IC50 | 2 | — | |
KEUZGQNTDMYNJZ
|
6.1 | IC50 | 2 | — |