Target Details
| UniProt AC | Q9BYW2 |
|---|---|
| Gene Symbol | SETD2 |
| Protein Name | Histone-lysine N-methyltransferase SETD2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF17907 (AWS) PF00856 (SET) PF08236 (SRI) PF00397 (WW) |
Summary
- Multi-target molecules 6
- Clinical molecules 0
- Avg pChEMBL 7.34
KEGG Pathways (2)
Associated Diseases (3)
Active Molecules (6)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZLVKIBLQXFILMA
|
7.9 | IC50 | 2 | — | |
ZNRYMFGQJYWIRE
|
7.8 | IC50 | 2 | — | |
PGNLXEBQMQHFNK
|
7.6 | IC50 | 2 | — | |
AAAQFGUYHFJNHI
|
7.3 | IC50 | 252 | — | |
GBIAQCRLFDZGOQ
|
7.2 | IC50 | 2 | — | |
IYOJRUQOOVAGRU
|
6.2 | IC50 | 2 | — |