Target Details
| UniProt AC | Q9BY41 |
|---|---|
| Gene Symbol | HDAC8 |
| Protein Name | Histone deacetylase 8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00850 (Hist_deacetyl) |
Summary
- Multi-target molecules 2,947
- Clinical molecules 486
- Avg pChEMBL 6.92
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (2,947)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NSHZNBNGZXAAFX
|
7.4 | IC50 | 11 | — | |
PHUXESRMVBVOSF
|
7.4 | IC50 | 11 | — | |
WFVUNJKMHRPDBB
|
7.4 | IC50 | 12 | Yes | |
WJUZCSPLBDPMTN
|
7.4 | IC50 | 3 | — | |
AIBMQRSNQIFQAL
|
7.4 | IC50 | 11 | Yes | |
BGPNDFOLJOUNJE
|
7.4 | IC50 | 11 | — | |
BKTQCQFRBAQVAT
|
7.4 | IC50 | 3 | — | |
LLXLAAHCAZIAKN
|
7.4 | IC50 | 11 | — | |
LZDVZSHIAKMDMZ
|
7.4 | IC50 | 4 | — | |
NDFSNVFVPNHHLM
|
7.4 | IC50 | 11 | — | |
PLNPDHQHVIPIPU
|
7.4 | IC50 | 3 | — | |
UMVVIIYGNDFZHN
|
7.4 | IC50 | 11 | — | |
WRXIPQCKJYKVSR
|
7.4 | IC50 | 11 | Yes | |
XSEMMBSLRMCHPX
|
7.4 | IC50 | 2 | — | |
GLUNWMQGDQEBAS
|
7.4 | IC50 | 12 | — | |
NUVBVOUKGLEFEW
|
7.4 | IC50 | 11 | — | |
XAISOELXZHHCPI
|
7.4 | IC50 | 2 | — | |
CKKPUWGKABSEIP
|
7.4 | IC50 | 4 | — | |
GYMSRUYUXJKIQR
|
7.4 | IC50 | 4 | — | |
HWSBOLCZWNNRGV
|
7.4 | IC50 | 11 | — | |
JZLYRFASZIDDDD
|
7.4 | IC50 | 11 | — | |
MCSQEIIMKDGXTR
|
7.4 | IC50 | 12 | Yes | |
PDJURBSVOZANDU
|
7.4 | IC50 | 6 | — | |
QBAGBBYBQAYFBT
|
7.4 | IC50 | 12 | Yes | |
RAZZTINTVZDPBL
|
7.4 | IC50 | 11 | — | |
RQBYQWASRFBDRN
|
7.4 | IC50 | 12 | Yes | |
RREMAKLSNSMREF
|
7.4 | IC50 | 4 | — | |
RXBHCXGBRWOPIP
|
7.4 | IC50 | 5 | — | |
SYKXAFABQPXBGT
|
7.4 | IC50 | 11 | — | |
VNRCXPZNHIIBGH
|
7.4 | IC50 | 5 | — | |
VZROKPBSFBHVTL
|
7.4 | IC50 | 12 | Yes | |
DANQOBBFZRKLFG
|
7.3 | IC50 | 11 | — | |
KXWBUKMWZKTHCV
|
7.3 | IC50 | 11 | — | |
SKZFNTOJPSTVDI
|
7.3 | IC50 | 4 | — | |
VADNNPZELPREQB
|
7.3 | IC50 | 11 | — | |
AFLGXRAIHNMVAQ
|
7.3 | IC50 | 11 | — | |
DOBGCSDZOYQKSP
|
7.3 | IC50 | 3 | — | |
LZCMBRQLXVTLOY
|
7.3 | IC50 | 12 | Yes | |
MXWDSZWTBOCWBK
|
7.3 | IC50 | 13 | Yes | |
QVOOYKPJQVGLIJ
|
7.3 | IC50 | 11 | — | |
VVGBYNYCWGLRCF
|
7.3 | IC50 | 3 | — | |
XERRUFOXNBPZPF
|
7.3 | IC50 | 11 | — | |
AZTHAJKEPBKWIZ
|
7.3 | IC50 | 3 | — | |
DTNVLAIWDVXDJR
|
7.3 | IC50 | 6 | — | |
GXSIKRXDVVRPGS
|
7.3 | IC50 | 11 | — | |
JXKIBHDACODLNS
|
7.3 | IC50 | 11 | — | |
MUMLRNZRMHNDNB
|
7.3 | IC50 | 11 | — | |
SCFMSNTXMREOOX
|
7.3 | IC50 | 4 | — | |
WGUXKEANCBSTED
|
7.3 | IC50 | 4 | — | |
YOJHPSLHBFFDDL
|
7.3 | IC50 | 19 | — |