Target Details
| UniProt AC | Q9BY41 |
|---|---|
| Gene Symbol | HDAC8 |
| Protein Name | Histone deacetylase 8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00850 (Hist_deacetyl) |
Summary
- Multi-target molecules 2,947
- Clinical molecules 486
- Avg pChEMBL 6.92
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (2,947)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XJRZGSQLQPWVJK
|
7.6 | IC50 | 3 | — | |
MEJLVLMAJJRLCR
|
7.6 | IC50 | 9 | Yes | |
MEJLVLMAJJRLCR
|
7.6 | IC50 | 7 | Yes | |
VPPDBLLRRNCUSU
|
7.6 | IC50 | 12 | — | |
DLBZBSURVFVXPO
|
7.6 | IC50 | 3 | — | |
JHAWARWGHKZRPV
|
7.6 | IC50 | 12 | — | |
JJOOKDGBBREJDT
|
7.6 | IC50 | 3 | — | |
NNVFBEZKIQPVJI
|
7.6 | IC50 | 11 | — | |
OHFSXIKHOCGMKB
|
7.6 | IC50 | 11 | — | |
PKADKDXQOLJENK
|
7.6 | IC50 | 12 | — | |
WTGMUNCNXTUDSC
|
7.6 | IC50 | 3 | — | |
ASHPRZYGCOMVHO
|
7.6 | IC50 | 3 | — | |
BEDWKBWRNPJVER
|
7.6 | IC50 | 11 | — | |
BVQUNILVJJVJFX
|
7.6 | IC50 | 11 | — | |
LNVJSKBRJGXMLU
|
7.6 | IC50 | 11 | — | |
NKOAGBYPCCDVOF
|
7.6 | IC50 | 4 | — | |
OGAKAZXENWFQRT
|
7.6 | IC50 | 12 | Yes | |
PIGOQJKXERKEJZ
|
7.6 | IC50 | 2 | — | |
VLJAVCKTTLIBDT
|
7.6 | IC50 | 4 | — | |
VPTVCYOEECUFBP
|
7.6 | IC50 | 4 | — | |
XJWSRFRYWHJEHD
|
7.6 | IC50 | 11 | — | |
XRHLECJNJSLFEN
|
7.6 | IC50 | 6 | — | |
XVUVRYUDMFGFHP
|
7.6 | IC50 | 11 | — | |
YBRAQRNYXSMWJX
|
7.6 | IC50 | 11 | — | |
USOAUSIBPGPBGY
|
7.6 | IC50 | 11 | — | |
CRAMEMOEGDTUCY
|
7.5 | IC50 | 11 | — | |
HUACOPNZWJZPLY
|
7.5 | IC50 | 11 | — | |
JSVSHZALVLCLJD
|
7.5 | IC50 | 11 | — | |
JXKKJJUGFLVTAG
|
7.5 | IC50 | 4 | — | |
SZDMMLKTDJTENB
|
7.5 | IC50 | 5 | — | |
VGDKNUOQFCSMED
|
7.5 | IC50 | 7 | — | |
WHZVNACXBWBBAT
|
7.5 | IC50 | 11 | — | |
YIQVYQNMHZMEBO
|
7.5 | IC50 | 4 | — | |
CCCCPSHFLXQUBH
|
7.5 | IC50 | 12 | — | |
CLPFHLPEOTXHDL
|
7.5 | IC50 | 12 | — | |
GKSYBLDJZMIKQE
|
7.5 | IC50 | 12 | — | |
GXYPZZICISCPIH
|
7.5 | IC50 | 4 | — | |
KQVHAPWDDOGVTF
|
7.5 | IC50 | 11 | — | |
NJJWVVQDXRGHLI
|
7.5 | IC50 | 11 | — | |
VJPAKRBNAKWZCJ
|
7.5 | IC50 | 11 | — | |
WTHQHAZITISKDC
|
7.5 | IC50 | 4 | — | |
JAEMGHJLPFENAA
|
7.5 | IC50 | 11 | — | |
NBHWQUHEYOFBKG
|
7.5 | IC50 | 11 | — | |
PKUNUWVORBBOHE
|
7.5 | IC50 | 12 | Yes | |
BKQJCMOVBFAIQR
|
7.5 | IC50 | 12 | Yes | |
BQUAPLIHVAVSDU
|
7.5 | IC50 | 12 | Yes | |
CITNMKKLNPYCDV
|
7.5 | IC50 | 11 | Yes | |
FGYOOZLOHGPAER
|
7.5 | IC50 | 3 | — | |
HMMNPRYLJPCLFS
|
7.5 | IC50 | 11 | — | |
IJBHQQMTDZNJTA
|
7.5 | IC50 | 11 | — |