Target Details
| UniProt AC | Q9BXF3 |
|---|---|
| Gene Symbol | CECR2 |
| Protein Name | Chromatin remodeling regulator CECR2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00439 (Bromodomain) |
Summary
- Multi-target molecules 48
- Clinical molecules 0
- Avg pChEMBL 6.87
KEGG Pathways (1)
Active Molecules (48)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RBUYFHLQNPJMQM
|
8.1 | Kd | 10 | — | |
MSIJJXOWLFOYIN
|
8.0 | Kd | 2 | — | |
QFRIGJQJVRCBFQ
|
8.0 | IC50 | 3 | — | |
UYBRROMMFMPJAN
|
8.0 | IC50 | 8 | — | |
CBGFEMSXMIJQKG
|
8.0 | IC50 | 3 | — | |
OWQNTPSDYOZXJM
|
8.0 | IC50 | 2 | — | |
UOQAFGWMKNIVAR
|
8.0 | Kd | 6 | — | |
RLNJZBANHSVNDS
|
7.9 | IC50 | 2 | — | |
ZKIRTFGYQVXNGL
|
7.8 | IC50 | 2 | — | |
ICIIHYCMSRJMHI
|
7.8 | IC50 | 2 | — | |
DBLNLPCEKQBLAI
|
7.7 | IC50 | 3 | — | |
IFILOJYOQZJYIC
|
7.7 | IC50 | 2 | — | |
KPWWFNXRLAAREN
|
7.4 | Kd | 12 | — | |
JYTISQGEFSHUIR
|
7.2 | Kd | 4 | — | |
HVFFRODVHZGRAZ
|
7.1 | IC50 | 4 | — | |
CHEXYSJBKQQXIF
|
7.1 | IC50 | 2 | — | |
AZCFROYDWGJIHI
|
7.0 | IC50 | 3 | — | |
VNCNIMOILJQAGJ
|
7.0 | IC50 | 2 | — | |
BJFSUDWKXGMUKA
|
6.9 | Kd | 3 | — | |
KWKAHJNKXUKKKE
|
6.9 | IC50 | 2 | — | |
XHAYAQCABOVSNX
|
6.9 | IC50 | 2 | — | |
PGRPAJVQVRBFEA
|
6.9 | IC50 | 2 | — | |
MYFFGZYMLKZBPZ
|
6.8 | IC50 | 4 | — | |
SPSRAFOXVSNAJA
|
6.8 | IC50 | 3 | — | |
WRUWGLUCNBMGPS
|
6.7 | IC50 | 5 | — | |
WZSQCCTZFYLIKW
|
6.6 | IC50 | 2 | — | |
YHMNROQTPUKNLA
|
6.6 | IC50 | 8 | — | |
DBZGKTULFWRCIP
|
6.6 | IC50 | 2 | — | |
XHAYAQCABOVSNX
|
6.6 | IC50 | 9 | — | |
YRWXMRVZJRZZNB
|
6.6 | IC50 | 2 | — | |
BQAKOVGAYWUDIT
|
6.4 | IC50 | 3 | — | |
MRADVJWFCVGIRG
|
6.4 | IC50 | 2 | — | |
RJEMCUZKQLRUIS
|
6.4 | IC50 | 4 | — | |
IHZXYEFDJOXHGJ
|
6.3 | IC50 | 2 | — | |
XSDOLOPLLGGSCB
|
6.3 | IC50 | 2 | — | |
ZACGKNYCBHUCNI
|
6.3 | IC50 | 2 | — | |
CMTGUEFAXALUTH
|
6.3 | IC50 | 3 | — | |
JIYPVUCBRQNICX
|
6.2 | Kd | 7 | — | |
KWYIXQZKANFDQR
|
6.2 | IC50 | 2 | — | |
BTTCKSLDCMBUAH
|
6.1 | Ki | 7 | — | |
POICMTYCJMMADL
|
6.1 | IC50 | 3 | — | |
QAORWPLEPWLSPU
|
6.1 | IC50 | 2 | — | |
DGJREYHVQYZTEV
|
6.0 | Kd | 6 | — | |
APJDTDALQSVARU
|
6.0 | IC50 | 3 | — | |
AVBQIZYXLUVYRI
|
6.0 | IC50 | 2 | — | |
IPQLFXYRKFCCRJ
|
6.0 | IC50 | 2 | — | |
WHKOQEHRVJBOCH
|
6.0 | IC50 | 2 | — | |
YTQRBAXLTKDECT
|
6.0 | Ki | 5 | — |