Target Details
| UniProt AC | Q9BXA7 |
|---|---|
| Gene Symbol | TSSK1B |
| Protein Name | Testis-specific serine/threonine-protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 63
- Clinical molecules 5
- Avg pChEMBL 6.91
Active Molecules (63)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OEEGUWWPGAZRIJ
|
6.1 | Ki | 21 | — | |
SQXSMLLCDWJNAC
|
6.1 | Ki | 20 | — | |
XYZNKCSDQRKAFR
|
6.1 | Ki | 53 | — | |
YEHCNYAQEBQCCS
|
6.1 | Ki | 74 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JOIUJUJSHIHBDT
|
6.0 | Ki | 18 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
NFMGZVPRGVERNN
|
6.0 | Ki | 44 | — | |
NHHQJBCNYHBUSI
|
6.0 | Kd | 220 | — | |
UUWNXFJBBYAMDT
|
6.0 | Ki | 46 | — | |
WYOMXSAYYXBPMN
|
6.0 | Ki | 24 | — | |
XSRHBCYNCKAFKS
|
6.0 | Ki | 45 | — |