Target Details
| UniProt AC | Q9BXA7 |
|---|---|
| Gene Symbol | TSSK1B |
| Protein Name | Testis-specific serine/threonine-protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 63
- Clinical molecules 5
- Avg pChEMBL 6.91
Active Molecules (63)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
10.2 | IC50 | 408 | — | |
IUWWRSQCDUQDEZ
|
9.7 | IC50 | 8 | — | |
IUWWRSQCDUQDEZ
|
9.7 | IC50 | 9 | — | |
AILRADAXUVEEIR
|
8.4 | IC50 | 75 | — | |
BSFNGHCTZDCQBF
|
8.2 | Ki | 93 | — | |
OWRXHGAFWZFFCW
|
8.1 | Ki | 113 | — | |
XPHWIERLJBFPFV
|
7.8 | Ki | 69 | — | |
NXSJMRCTGYTSTK
|
7.7 | Kd | 200 | — | |
OSVUGUHRKMMBSE
|
7.7 | Kd | 170 | — | |
UEFCSGDOOJJXTN
|
7.7 | IC50 | 46 | — | |
VERWOWGGCGHDQE
|
7.6 | IC50 | 23 | — | |
HKSZLNNOFSGOKW
|
7.6 | Kd | 213 | — | |
QQWUGDVOUVUTOY
|
7.6 | Kd | 231 | Yes | |
MVJMMLFMPWITEJ
|
7.5 | Ki | 110 | — | |
UMTWTCVTRDYHQQ
|
7.5 | Ki | 56 | — | |
BNSPEWBMGVWZFC
|
7.5 | IC50 | 7 | — | |
RYYNGWLOYLRZLK
|
7.3 | Ki | 104 | — | |
YOVNFNXUCOWYSG
|
7.3 | Ki | 33 | Yes | |
ADMFLILDQJSEIK
|
7.2 | Ki | 72 | — | |
CKVWQORGCCEYHS
|
7.2 | Ki | 50 | — | |
JZTOUVBEZONDKA
|
7.1 | Ki | 80 | — | |
PCQMERRARZKTPW
|
7.1 | Ki | 68 | — | |
UIARLYUEJFELEN
|
7.0 | Kd | 289 | Yes | |
CHTMRWQLNNRRFJ
|
7.0 | Ki | 70 | — | |
NJPWCTYVEJIQBM
|
7.0 | Ki | 72 | — | |
FLEAYYMORDPWAJ
|
6.9 | Ki | 90 | — | |
FUMCKNCUEAQHCV
|
6.9 | Ki | 103 | — | |
UDFDIIVNIYWXDM
|
6.8 | Ki | 74 | — | |
AOBLBPWPSKBHSI
|
6.7 | Ki | 55 | — | |
GDYZFFBMSBDTAA
|
6.7 | Ki | 60 | — | |
JSKUWFIZUALZLX
|
6.7 | Ki | 33 | — | |
WINHZLLDWRZWRT
|
6.7 | Ki | 66 | — | |
XFWUTMHVDGPWLH
|
6.7 | Ki | 75 | — | |
DGLFSNZWRYADFC
|
6.7 | IC50 | 12 | — | |
LRZYYIZFBXFSJB
|
6.6 | Ki | 69 | — | |
MASJMHFQMYAPJR
|
6.6 | Ki | 41 | — | |
RJZDECGDCKOHBV
|
6.6 | Ki | 70 | — | |
VXYDJXMHISGSDA
|
6.6 | Ki | 59 | — | |
GCYXEGSPUDSZJY
|
6.5 | Ki | 82 | — | |
HZTYDQRUAWIZRE
|
6.3 | Kd | 40 | Yes | |
HEUSUIRCBWROMH
|
6.3 | Ki | 64 | — | |
PIQCTGMSNWUMAF
|
6.3 | Ki | 137 | Yes | |
SBFPHSVZEXSHTL
|
6.3 | Ki | 62 | — | |
XKFTZKGMDDZMJI
|
6.3 | Ki | 56 | — | |
YWTBGJGMTBHQTM
|
6.3 | Ki | 65 | — | |
BPNUQXPIQBZCMR
|
6.2 | Ki | 60 | — | |
PSCJSWRVCKUMSL
|
6.2 | Ki | 35 | — | |
UVZVWLFSZNPMBS
|
6.2 | Ki | 17 | — | |
YUOWJICKAJQZLS
|
6.2 | Ki | 35 | — | |
GQLWKGVBOIYMTN
|
6.1 | Ki | 35 | — |