Target Details
| UniProt AC | Q9BVS4 |
|---|---|
| Gene Symbol | RIOK2 |
| Protein Name | Serine/threonine-protein kinase RIO2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01163 (RIO1) PF09202 (Rio2_N) |
Summary
- Multi-target molecules 17
- Clinical molecules 6
- Avg pChEMBL 6.43
KEGG Pathways (1)
Active Molecules (17)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WINHZLLDWRZWRT
|
7.3 | Kd | 201 | Yes | |
BMGQWWVMWDBQGC
|
7.0 | Kd | 147 | Yes | |
CTNPALGJUAXMMC
|
6.8 | Kd | 151 | — | |
HPQZTEVMVAVGJO
|
6.8 | Kd | 5 | — | |
CYLDJPVEBVIXNB
|
6.6 | Kd | 6 | — | |
GCIKSSRWRFVXBI
|
6.6 | Kd | 109 | Yes | |
PIQCTGMSNWUMAF
|
6.6 | Kd | 137 | Yes | |
HKSZLNNOFSGOKW
|
6.4 | Kd | 408 | — | |
ODPGGGTTYSGTGO
|
6.3 | Kd | 153 | — | |
CUIHSIWYWATEQL
|
6.2 | Kd | 61 | Yes | |
YBXRSCXGRPSTMW
|
6.2 | Kd | 6 | — | |
LHNIIDJUOCFXAP
|
6.2 | Kd | 20 | Yes | |
TUVCWJQQGGETHL
|
6.1 | Kd | 22 | — | |
YZDJQTHVDDOVHR
|
6.1 | Kd | 23 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |