Target Details
| UniProt AC | Q9BUB5 |
|---|---|
| Gene Symbol | MKNK1 |
| Protein Name | MAP kinase-interacting serine/threonine-protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 445
- Clinical molecules 13
- Avg pChEMBL 7.24
KEGG Pathways (3)
Active Molecules (445)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GFNNBHLJANVSQV
|
6.3 | IC50 | 7 | Yes | |
GVZURVVGRNHCLH
|
6.3 | IC50 | 2 | — | |
HRLBMFYCQTZRNE
|
6.3 | IC50 | 2 | — | |
LZDLAOSZVOKASQ
|
6.3 | IC50 | 2 | — | |
MCHMLUWPNDLLEY
|
6.3 | IC50 | 2 | — | |
GFYFRPOVKHGTOX
|
6.3 | IC50 | 2 | — | |
HXNIAYXLNXQQOW
|
6.3 | IC50 | 2 | — | |
PGCQCLPSSJBTRH
|
6.3 | IC50 | 2 | — | |
PLZBJLWXNDHFTE
|
6.3 | IC50 | 2 | — | |
XOAMVMHKXHJDNZ
|
6.3 | IC50 | 2 | — | |
ZEQJVQLQTLNOBZ
|
6.3 | IC50 | 2 | — | |
PFHIDQUYVRCLAG
|
6.2 | IC50 | 2 | — | |
UXNUQVZRIJPJBL
|
6.2 | IC50 | 2 | — | |
OGNWKFYJHNZTNC
|
6.2 | IC50 | 2 | — | |
AJSPQFHUVJMVLQ
|
6.2 | IC50 | 2 | — | |
OCBKWOSSKSMBOO
|
6.2 | IC50 | 2 | — | |
LSPANGZZENHZNJ
|
6.2 | IC50 | 10 | Yes | |
HWKLPUXMYLCSIE
|
6.2 | IC50 | 2 | — | |
VXNHTGWDWVCFSI
|
6.2 | IC50 | 2 | — | |
XFFNHXOXHSUYQQ
|
6.2 | IC50 | 2 | — | |
DKRBCZRLAIEHLG
|
6.2 | IC50 | 2 | — | |
FKCRUIWBTDNJFG
|
6.2 | IC50 | 4 | — | |
IEPPUFLBHOABDC
|
6.2 | IC50 | 2 | — | |
AAKJLRGGTJKAMG
|
6.2 | Kd | 50 | Yes | |
DXSFSGMRGCIRSG
|
6.2 | IC50 | 2 | — | |
KAZFNRNYKKXSJQ
|
6.2 | IC50 | 2 | — | |
PZNMULIOTSQSJK
|
6.2 | IC50 | 2 | — | |
NOZFCTAJFMLWPE
|
6.2 | IC50 | 2 | — | |
TUPFDIJWABCYHK
|
6.2 | Ki | 2 | — | |
MUFGPGISRVJPDN
|
6.1 | IC50 | 2 | — | |
NLOCXNJSWCSWJT
|
6.1 | IC50 | 2 | — | |
BKIZDYJBKOZFQS
|
6.1 | IC50 | 2 | — | |
LLDMEDJNOJVTEE
|
6.1 | IC50 | 2 | — | |
YBOOAZFLAUPOKA
|
6.1 | Ki | 3 | — | |
DZEKKRSPIVXYAJ
|
6.1 | IC50 | 2 | — | |
IBHOTNCJTRATHT
|
6.1 | IC50 | 2 | — | |
LPDCQOLOXLFVBW
|
6.1 | IC50 | 2 | — | |
UJIAQDJKSXQLIT
|
6.1 | Kd | 38 | — | |
UQPMANVRZYYQMD
|
6.1 | IC50 | 3 | — | |
ABOJMONYYGQPBY
|
6.0 | IC50 | 2 | — | |
DUVXFOSLZHSJPX
|
6.0 | Ki | 3 | — | |
WLLDFEGKGAPLQO
|
6.0 | IC50 | 2 | — | |
JZBMRMXXSMSEAY
|
6.0 | IC50 | 2 | — | |
QVHDOESZFDSEKS
|
6.0 | Ki | 2 | — | |
RELLPRKUGXVDBP
|
6.0 | Ki | 2 | — |