Target Details
| UniProt AC | Q9BUB5 |
|---|---|
| Gene Symbol | MKNK1 |
| Protein Name | MAP kinase-interacting serine/threonine-protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 445
- Clinical molecules 13
- Avg pChEMBL 7.24
KEGG Pathways (3)
Active Molecules (445)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZROBKNPXIOQRBD
|
6.5 | IC50 | 2 | — | |
XGALLCVXEZPNRQ
|
6.5 | Kd | 39 | Yes | |
XJFORULEXOZBAQ
|
6.5 | IC50 | 2 | — | |
TWYKNRDHNFNBDF
|
6.5 | IC50 | 2 | — | |
HSJFJXIKCSINLE
|
6.5 | Ki | 2 | — | |
LKFLRBIQIXBCCO
|
6.5 | IC50 | 2 | — | |
IMLMBHVOASBVOW
|
6.5 | IC50 | 2 | — | |
RVMLNNCKNCFOFH
|
6.5 | IC50 | 4 | — | |
RYUUMGNHANZHLX
|
6.5 | Ki | 2 | — | |
QXPNJMHRUZCEAP
|
6.5 | IC50 | 14 | — | |
FRWDDDSGEGTXIY
|
6.5 | IC50 | 2 | — | |
KKUMLZFCIPKXAO
|
6.5 | IC50 | 2 | — | |
ZDSCMCRGHRMVAM
|
6.5 | IC50 | 2 | — | |
GHOGNCOJXOPHJS
|
6.5 | IC50 | 2 | — | |
VFSUAKYNPKYPLY
|
6.5 | Ki | 2 | — | |
ANUKWIYBPKFKPT
|
6.5 | IC50 | 2 | — | |
SIILILXNZLEIIT
|
6.5 | IC50 | 2 | — | |
UHTHHESEBZOYNR
|
6.4 | Kd | 66 | Yes | |
ZAUQVEIJQHLVAR
|
6.4 | IC50 | 2 | — | |
ZBOZMNJGIZGSFL
|
6.4 | IC50 | 2 | — | |
FEXHRQNJTUVDQQ
|
6.4 | IC50 | 2 | — | |
PQAKQADTDVGYOC
|
6.4 | IC50 | 2 | — | |
UKTICNMOUVEYRR
|
6.4 | IC50 | 4 | — | |
ZLXQWGHPSCNGQC
|
6.4 | IC50 | 2 | — | |
FETVSVYRUZPIRW
|
6.4 | IC50 | 2 | — | |
LJNQZRKFYXYCCW
|
6.4 | IC50 | 2 | — | |
YLNVYSOHEOBKJW
|
6.4 | IC50 | 2 | — | |
JSXSJAZHNLZZFG
|
6.4 | IC50 | 2 | — | |
SQBBTXGGRJHRGB
|
6.4 | IC50 | 2 | — | |
HIPFDFQYWKJHND
|
6.4 | IC50 | 2 | — | |
QRDADMUYUNCQDD
|
6.4 | IC50 | 2 | — | |
SGVAIMLQDSZAQH
|
6.4 | IC50 | 2 | — | |
SSHPOTBZTFBVDB
|
6.4 | IC50 | 2 | — | |
FYKZPCLKTZZIBA
|
6.4 | IC50 | 2 | — | |
MYUBZXFNNULBFX
|
6.4 | IC50 | 2 | — | |
YXYNMHMVPRQKBT
|
6.4 | IC50 | 2 | — | |
HKOAGBQDHYMZTP
|
6.3 | IC50 | 2 | — | |
OJASUOZKOQBQAR
|
6.3 | IC50 | 2 | — | |
VTNHUNPWAHGVCA
|
6.3 | IC50 | 2 | — | |
GMAZHMAIHCELNK
|
6.3 | IC50 | 2 | — | |
UUVPHDJCRCLZOZ
|
6.3 | IC50 | 2 | — | |
UXIRCXIRZUXJSJ
|
6.3 | IC50 | 2 | — | |
QHPJIUARPKBLQQ
|
6.3 | IC50 | 3 | — | |
LXZQZRCDEXIVBU
|
6.3 | IC50 | 2 | — | |
QUFSPIHVCCPJER
|
6.3 | IC50 | 2 | — | |
SHKWWTGWEWLIRC
|
6.3 | IC50 | 2 | — | |
VUQPNTNKEPWYRO
|
6.3 | IC50 | 2 | — | |
FCCJIRJUDAWXRO
|
6.3 | IC50 | 4 | — | |
GCTFTMWXZFLTRR
|
6.3 | IC50 | 7 | — | |
GEWLYFZWVLXQME
|
6.3 | Ki | 2 | — |