Target Details
| UniProt AC | Q9BUB5 |
|---|---|
| Gene Symbol | MKNK1 |
| Protein Name | MAP kinase-interacting serine/threonine-protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 445
- Clinical molecules 13
- Avg pChEMBL 7.24
KEGG Pathways (3)
Active Molecules (445)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UAPCOTPXNOKKFY
|
6.9 | IC50 | 2 | — | |
GHOGNCOJXOPHJS
|
6.8 | IC50 | 2 | — | |
PTSMJMBYLZTCHZ
|
6.8 | IC50 | 2 | — | |
QKBPOTWGKPRFEH
|
6.8 | IC50 | 2 | — | |
UTOQFKLQNHKULZ
|
6.8 | Ki | 2 | — | |
JPWNVOHBTSBREO
|
6.8 | IC50 | 2 | — | |
HIIXSKLGSBCTAH
|
6.8 | IC50 | 3 | — | |
LKQCQDSSPGVMPT
|
6.8 | IC50 | 2 | — | |
RKAHOQATMSONTM
|
6.8 | IC50 | 6 | — | |
TXTJPVXASVJOMW
|
6.8 | IC50 | 2 | — | |
CWROOQSMUQCFMV
|
6.8 | IC50 | 2 | — | |
DYIZARYDRMKISJ
|
6.8 | IC50 | 2 | — | |
HEPDAJRNJBNJAE
|
6.8 | IC50 | 15 | Yes | |
OOKMVSGWNLPFAW
|
6.8 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
6.8 | Kd | 213 | — | |
XEPPZNCGRACPGZ
|
6.8 | IC50 | 2 | — | |
JONUUBFCZUAOFY
|
6.8 | IC50 | 10 | — | |
CQJWUWZZQUEKGG
|
6.7 | IC50 | 2 | — | |
DITKYYZRIWWAQK
|
6.7 | IC50 | 2 | — | |
NGBWQVJCOYTGOR
|
6.7 | IC50 | 8 | — | |
WZDDWQHGNFSHRU
|
6.7 | IC50 | 2 | — | |
CRQZRBXFLRRAIQ
|
6.7 | Ki | 2 | — | |
HINOQCZIDBNXEI
|
6.7 | IC50 | 5 | — | |
MCHMLUWPNDLLEY
|
6.7 | IC50 | 2 | — | |
CGMQSJXTBXHOTH
|
6.7 | IC50 | 9 | — | |
FXMBSEOFWALADX
|
6.7 | IC50 | 3 | — | |
GHOGNCOJXOPHJS
|
6.7 | IC50 | 2 | — | |
YIHNQOZIZBZUOT
|
6.7 | IC50 | 2 | — | |
ZJWPYYIRORJZPQ
|
6.7 | IC50 | 4 | — | |
OISBNGXKBOCXER
|
6.7 | IC50 | 2 | — | |
RRSGLFRYYGSFFX
|
6.7 | IC50 | 2 | — | |
SQGZUMNITNRRET
|
6.7 | IC50 | 2 | — | |
WZILQEFHQBNHBB
|
6.7 | IC50 | 2 | — | |
ZIOVJRQVOJIVAE
|
6.7 | IC50 | 2 | — | |
KOGDOKSJNXRDBX
|
6.7 | IC50 | 2 | — | |
LPLVTTVTTDMYHT
|
6.7 | IC50 | 2 | — | |
KJZWOUQMPQCYIK
|
6.7 | IC50 | 2 | — | |
MLDQJTXFUGDVEO
|
6.6 | Kd | 85 | Yes | |
NHHQJBCNYHBUSI
|
6.6 | Kd | 220 | — | |
ZJBOENMAUCUUIV
|
6.6 | IC50 | 2 | — | |
LJQCFLSZUSTALC
|
6.6 | IC50 | 2 | — | |
OWXKIXPMTVEDCR
|
6.6 | IC50 | 2 | — | |
RKBMAROJKLHAMI
|
6.6 | IC50 | 6 | — | |
XGWSCBXZMXUGRN
|
6.6 | IC50 | 2 | — | |
FDYURKPWOPRSMM
|
6.6 | IC50 | 2 | — | |
OMZCMEYTWSXEPZ
|
6.6 | Kd | 43 | Yes | |
HVHRHDHQHUAOQI
|
6.6 | IC50 | 5 | — | |
XPBVTQGDRIYCRN
|
6.6 | IC50 | 2 | — | |
LFEOCNIHNYNYIJ
|
6.5 | IC50 | 2 | — | |
OJGVXOPNHCRTAD
|
6.5 | IC50 | 2 | — |