Target Details
| UniProt AC | Q9BUB5 |
|---|---|
| Gene Symbol | MKNK1 |
| Protein Name | MAP kinase-interacting serine/threonine-protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 445
- Clinical molecules 13
- Avg pChEMBL 7.24
KEGG Pathways (3)
Active Molecules (445)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LDVFAQGTHMKMLC
|
7.2 | IC50 | 2 | — | |
CXQHYVUVSFXTMY
|
7.1 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
7.1 | Kd | 149 | — | |
LCQIIAREQLPINL
|
7.1 | IC50 | 2 | — | |
VCSAIKGXBLLWTR
|
7.1 | IC50 | 2 | — | |
CWUHWURRJXDZRD
|
7.1 | Ki | 2 | — | |
FKXRAFMZZZCZIC
|
7.1 | IC50 | 2 | — | |
YHFVWRQJZMNUCR
|
7.1 | IC50 | 2 | — | |
OYOKXIIAQLUGEQ
|
7.1 | IC50 | 2 | — | |
CBAKEHNEEJTUGB
|
7.1 | IC50 | 2 | — | |
OPCZBBDJOVZICW
|
7.1 | IC50 | 2 | — | |
RCCFIMHYOFIWHJ
|
7.1 | IC50 | 2 | — | |
SIRSNKXGOCRFCT
|
7.1 | IC50 | 2 | — | |
PDEDJMZPQFJDNA
|
7.1 | IC50 | 2 | — | |
RLLAJTFWKAYWBI
|
7.1 | IC50 | 2 | — | |
SRVMCTQCWVQBNL
|
7.1 | IC50 | 2 | — | |
AILRADAXUVEEIR
|
7.1 | IC50 | 75 | — | |
JFZYWAILFVBGGL
|
7.1 | IC50 | 2 | — | |
VKRHDQYSQQELAD
|
7.0 | IC50 | 2 | — | |
ILYKJXYOFZKJGR
|
7.0 | IC50 | 2 | — | |
RKDUDJILSVKJSN
|
7.0 | IC50 | 2 | — | |
WVIQCXQWRJXXGZ
|
7.0 | IC50 | 2 | — | |
ZDNCMUXDGZVSHU
|
7.0 | IC50 | 2 | — | |
CARBAQLLNJEQRM
|
7.0 | IC50 | 2 | — | |
DPPHWOJYKINIBO
|
7.0 | IC50 | 2 | — | |
GHOGNCOJXOPHJS
|
7.0 | IC50 | 2 | — | |
LXOPXNJLPKCVBS
|
7.0 | IC50 | 2 | — | |
OHEKKVOQVJUAQW
|
7.0 | IC50 | 2 | — | |
PXYXJSKWHPGJFP
|
7.0 | IC50 | 2 | — | |
RNWLWPQNWGNPLV
|
7.0 | IC50 | 2 | — | |
GUXLMYYFWLSMCP
|
7.0 | IC50 | 2 | — | |
HNWUOUYCKCPSHE
|
7.0 | IC50 | 2 | — | |
JMVDIGHUQAXWIE
|
7.0 | IC50 | 10 | — | |
MLNZVQPAJITTGP
|
7.0 | IC50 | 2 | — | |
ZGXLPGBXVQLLJW
|
7.0 | Ki | 2 | — | |
GNLVXKVGJVMDRM
|
7.0 | IC50 | 2 | — | |
ALRLENDIHGVVDY
|
6.9 | IC50 | 2 | — | |
KQODTAOSMRHZLK
|
6.9 | IC50 | 2 | — | |
CLRWMPFUTCKUQH
|
6.9 | IC50 | 3 | — | |
DGUSKGFGXIHXKS
|
6.9 | IC50 | 2 | — | |
KAVINHSQSZLJGI
|
6.9 | IC50 | 2 | — | |
MYKOWOGZBMOVBJ
|
6.9 | IC50 | 9 | — | |
ZVSNSFQQKSZZMY
|
6.9 | IC50 | 7 | — | |
GQPLXSNGJYAHSH
|
6.9 | IC50 | 3 | — | |
HMVSRLUUXHNABC
|
6.9 | IC50 | 2 | — | |
HZVIUNVVQJWYNZ
|
6.9 | IC50 | 2 | — | |
OWEDOBFUVPKBNA
|
6.9 | IC50 | 2 | — | |
FXUCGEVPOQUSIH
|
6.9 | IC50 | 2 | — | |
OOQJIJYKWXLQNC
|
6.9 | IC50 | 16 | Yes | |
HEBJJJVAANGHLJ
|
6.9 | IC50 | 2 | — |