Target Details
| UniProt AC | Q9BUB5 |
|---|---|
| Gene Symbol | MKNK1 |
| Protein Name | MAP kinase-interacting serine/threonine-protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 445
- Clinical molecules 13
- Avg pChEMBL 7.24
KEGG Pathways (3)
Active Molecules (445)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GAWJEBCHHUPVEO
|
7.3 | IC50 | 2 | — | |
GVYZOWDBQXKJDR
|
7.3 | IC50 | 2 | — | |
HHGUCXDDCLOWPZ
|
7.3 | IC50 | 2 | — | |
IUWQSSGZFYFDEM
|
7.3 | IC50 | 2 | — | |
JQJVPKQUOPODEZ
|
7.3 | IC50 | 2 | — | |
JVKICFJXJPDNOJ
|
7.3 | IC50 | 2 | — | |
JYJWZHLMBPNEJV
|
7.3 | IC50 | 2 | — | |
KLPWXPHBHLDCCS
|
7.3 | IC50 | 2 | — | |
KQXTVRJPONHNFY
|
7.3 | IC50 | 2 | — | |
LXZXQQXBXVENQD
|
7.3 | IC50 | 2 | — | |
MTMFRAIOFPWKIH
|
7.3 | IC50 | 2 | — | |
OLGSXYPPKJJNJR
|
7.3 | IC50 | 2 | — | |
OPZFLEPCEIJFSE
|
7.3 | IC50 | 2 | — | |
PVFRNMLGINKVRT
|
7.3 | IC50 | 2 | — | |
QIMGDBHWVXEGQS
|
7.3 | IC50 | 2 | — | |
RCEKLIVCBVRHEU
|
7.3 | IC50 | 2 | — | |
RJINHNWMTFJSBN
|
7.3 | IC50 | 2 | — | |
RSJWFQUCOMWKQD
|
7.3 | IC50 | 2 | — | |
SXKIBLJFZKDDCP
|
7.3 | IC50 | 2 | — | |
UDXGUYCTMQSGOM
|
7.3 | IC50 | 2 | — | |
VKZOMKUUMGEJLL
|
7.3 | IC50 | 2 | — | |
VMPOUPXTRIFPLU
|
7.3 | IC50 | 2 | — | |
YCHQXPNHRHYUIG
|
7.3 | IC50 | 2 | — | |
HUFOBMZPSQAJRA
|
7.2 | IC50 | 2 | — | |
IXQFWQXAZJXVSH
|
7.2 | IC50 | 2 | — | |
JTKZYIFZLHCCDD
|
7.2 | IC50 | 2 | — | |
UIARLYUEJFELEN
|
7.2 | Kd | 289 | Yes | |
FMNWOBLAZAYOSG
|
7.2 | IC50 | 5 | — | |
IGCYGNGFBOQMOJ
|
7.2 | IC50 | 2 | — | |
TVBANCDFRJJEKJ
|
7.2 | IC50 | 2 | — | |
CQPDKJQEKIKEFC
|
7.2 | IC50 | 2 | — | |
DFAUAZYINZOIAU
|
7.2 | IC50 | 2 | — | |
DWHJLJMQWMLRNN
|
7.2 | IC50 | 2 | — | |
KSAKIZZKHCPIFK
|
7.2 | IC50 | 2 | — | |
YUDKTFUCCPOVGR
|
7.2 | IC50 | 2 | — | |
HECFVRUHGZHVGD
|
7.2 | IC50 | 2 | — | |
KTBKRHUBYKAUFQ
|
7.2 | IC50 | 2 | — | |
ZBKQXBZXZYIRIU
|
7.2 | IC50 | 2 | — | |
WSLNKDCNHNOGHL
|
7.2 | IC50 | 3 | — | |
CRIJBFDDOUPGQZ
|
7.2 | IC50 | 2 | — | |
FWRFPHJSGLYXTD
|
7.2 | IC50 | 3 | — | |
LGXIHGFTIXRTGJ
|
7.2 | IC50 | 2 | — | |
YAVNDOLVFFVVBX
|
7.2 | IC50 | 2 | — | |
MWCAWBUYZQRAJP
|
7.2 | IC50 | 2 | — | |
OGLZUCMDAWETHK
|
7.2 | IC50 | 2 | — | |
VKHXISWCFPVDEJ
|
7.2 | IC50 | 2 | — | |
ZDXIDBRGTYDHBQ
|
7.2 | IC50 | 5 | — | |
RNFXZZCKTTUGHL
|
7.2 | IC50 | 2 | — | |
ZLSMBKJDRUZGNN
|
7.2 | IC50 | 2 | — | |
ZAYMIFRCEPHPHT
|
7.2 | IC50 | 2 | — |