Target Details
| UniProt AC | Q9BUB5 |
|---|---|
| Gene Symbol | MKNK1 |
| Protein Name | MAP kinase-interacting serine/threonine-protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 445
- Clinical molecules 13
- Avg pChEMBL 7.24
KEGG Pathways (3)
Active Molecules (445)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VKHXISWCFPVDEJ
|
7.4 | IC50 | 2 | — | |
CMDIADSAZCFCCT
|
7.4 | IC50 | 2 | — | |
HVXHSDUKHSDIIZ
|
7.4 | IC50 | 2 | — | |
KVGHGVHKZQAQLD
|
7.4 | IC50 | 3 | — | |
KVPRKFQTIYGEJA
|
7.4 | IC50 | 2 | — | |
KVPRKFQTIYGEJA
|
7.4 | IC50 | 2 | — | |
MCHMLUWPNDLLEY
|
7.4 | IC50 | 2 | — | |
MQLVVLKXNBHGDG
|
7.4 | IC50 | 2 | — | |
OVAFHXUOPSXQOF
|
7.4 | IC50 | 2 | — | |
UMMWOVSZRFTRPV
|
7.4 | IC50 | 2 | — | |
UUQZSFPVUKCRKO
|
7.4 | IC50 | 3 | — | |
YCJJNSYFXNUIAV
|
7.4 | IC50 | 2 | — | |
ASJBYMJMNYQSDB
|
7.4 | IC50 | 2 | — | |
MNORXFRHDOWTKB
|
7.4 | IC50 | 2 | — | |
CSOGCPCCVIPBIK
|
7.4 | IC50 | 2 | — | |
FWTDZBZYPAAGCF
|
7.4 | IC50 | 2 | — | |
GEWLYFZWVLXQME
|
7.4 | IC50 | 9 | — | |
UUUBVRVITMLFJU
|
7.4 | IC50 | 2 | — | |
AGTYIHYYCHWRMP
|
7.4 | IC50 | 2 | — | |
OPQXXINFFAZXDD
|
7.4 | IC50 | 2 | — | |
QCKSDSPCHDSAHA
|
7.3 | IC50 | 2 | — | |
WMXDIPVFXWNELM
|
7.3 | IC50 | 14 | Yes | |
WPRQIYVTQUOMGG
|
7.3 | IC50 | 2 | — | |
NMGPJZFKRNRWDG
|
7.3 | IC50 | 2 | — | |
BDNVJOGXLGPBFH
|
7.3 | IC50 | 2 | — | |
KBJGQQRVHPTDJO
|
7.3 | IC50 | 2 | — | |
ACCGDLRUTZSFSS
|
7.3 | IC50 | 2 | — | |
ACCGDLRUTZSFSS
|
7.3 | IC50 | 2 | — | |
CLIORPUQKOJRDE
|
7.3 | IC50 | 3 | — | |
DPFZKILBVWKIDP
|
7.3 | IC50 | 3 | — | |
FOQNSWUDBARUFL
|
7.3 | IC50 | 3 | — | |
FPQBGLUWBCLXFG
|
7.3 | IC50 | 3 | — | |
QUVIEDJGNUFDDH
|
7.3 | IC50 | 3 | — | |
CRNUXVFKYMTHAJ
|
7.3 | IC50 | 2 | — | |
DZCGBMMTMNQQHW
|
7.3 | IC50 | 2 | — | |
FSROQMVTCKZCAM
|
7.3 | IC50 | 2 | — | |
MOQHPHSZEODHGL
|
7.3 | IC50 | 2 | — | |
TZHJOOVYOQMSSP
|
7.3 | IC50 | 2 | — | |
WHDVHWQDQBHJEN
|
7.3 | IC50 | 2 | — | |
AHGFXLZWTGRAAT
|
7.3 | IC50 | 2 | — | |
CUSAZOGXBMLNCR
|
7.3 | IC50 | 2 | — | |
ZZONCZDKYUYGTE
|
7.3 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.3 | IC50 | 408 | — | |
TXTSSJDYULDSBL
|
7.3 | IC50 | 2 | — | |
UXHZMEYLBGGTQR
|
7.3 | IC50 | 2 | — | |
VFWWHCOMWRSXME
|
7.3 | IC50 | 2 | — | |
BMCIBDDLDCNKAP
|
7.3 | IC50 | 2 | — | |
DBLJVNGTXRPKMS
|
7.3 | IC50 | 2 | — | |
DXRIPNKUBZNZQN
|
7.3 | IC50 | 2 | — | |
FGFUUBCEERIDBQ
|
7.3 | IC50 | 2 | — |