Target Details
| UniProt AC | Q9BUB5 |
|---|---|
| Gene Symbol | MKNK1 |
| Protein Name | MAP kinase-interacting serine/threonine-protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 445
- Clinical molecules 13
- Avg pChEMBL 7.24
KEGG Pathways (3)
Active Molecules (445)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AFKOJENZZZUAJE
|
7.7 | IC50 | 2 | — | |
PEHQJHHHTXOGJK
|
7.7 | IC50 | 2 | — | |
NSJGELDCKSGQQG
|
7.7 | IC50 | 2 | — | |
RIYDOTWDTHRXAQ
|
7.7 | IC50 | 2 | — | |
UNFYWRADYYEYQC
|
7.7 | IC50 | 2 | — | |
LACOTCUHEDDNGC
|
7.7 | IC50 | 2 | — | |
PFYNAVHEBIAEKL
|
7.7 | IC50 | 2 | — | |
PYMYZZLESAPEGL
|
7.7 | IC50 | 2 | — | |
YRDRYCRFGSQZQW
|
7.7 | IC50 | 2 | — | |
WTCFYBGLEUOJNE
|
7.6 | IC50 | 2 | — | |
MOHKECCWMOAJNH
|
7.6 | IC50 | 2 | — | |
QUCVXIHKWBYLLK
|
7.6 | IC50 | 2 | — | |
DXBQRCVASKKRRR
|
7.6 | IC50 | 2 | — | |
GCMXEMBFFWKSQR
|
7.6 | IC50 | 2 | — | |
PJFYYYJFEHNOHR
|
7.6 | IC50 | 2 | — | |
XCQQKYFEUUGRAR
|
7.6 | IC50 | 2 | — | |
ODPGGGTTYSGTGO
|
7.6 | Kd | 153 | — | |
GRHDTNANZAYFHJ
|
7.6 | IC50 | 2 | — | |
JRKYKAKARRYSSS
|
7.6 | IC50 | 14 | Yes | |
SHFKCVNKUAWFOE
|
7.6 | IC50 | 2 | — | |
CHQYMHAUSYCZKU
|
7.6 | IC50 | 2 | — | |
CSOGCPCCVIPBIK
|
7.6 | IC50 | 2 | — | |
FOGVEYPAPSELLE
|
7.5 | IC50 | 2 | — | |
OXVAVDAJVDRCDN
|
7.5 | IC50 | 2 | — | |
PCPQKTHZHZRQEF
|
7.5 | IC50 | 2 | — | |
GKGFTCRWDLEQNT
|
7.5 | IC50 | 2 | — | |
IHHXSJUBRJFSFB
|
7.5 | IC50 | 2 | — | |
QHADVLVFMKEIIP
|
7.5 | IC50 | 9 | — | |
HJIRNKSTJOICTI
|
7.5 | IC50 | 2 | — | |
IOBRLFTZHXZWPT
|
7.5 | IC50 | 2 | — | |
XEUHVTVNJONCLA
|
7.5 | IC50 | 2 | — | |
TXLKAUPPLBUDKU
|
7.5 | IC50 | 2 | — | |
USRICZTXNXFJQE
|
7.5 | IC50 | 2 | — | |
VQBHHVIUAXNAOC
|
7.5 | IC50 | 2 | — | |
VQZTVBGPAZGVHT
|
7.5 | IC50 | 2 | — | |
MOUJAAFOCZZGAI
|
7.5 | IC50 | 2 | — | |
YFJVDNQENDFYRT
|
7.5 | IC50 | 2 | — | |
ZFJOWPQCUFNQSC
|
7.5 | IC50 | 2 | — | |
CJQYSYNGPPQQJW
|
7.5 | IC50 | 2 | — | |
RTSIVZFZSQNFQG
|
7.5 | IC50 | 2 | — | |
PCSNHSCJJFGAOB
|
7.4 | IC50 | 3 | — | |
TUWVKXVVEYHYAW
|
7.4 | IC50 | 2 | — | |
CDELWNRTTCPMLW
|
7.4 | IC50 | 2 | — | |
DHAZVVKQOCTFFZ
|
7.4 | IC50 | 2 | — | |
OGDZDXFTNNLXFS
|
7.4 | IC50 | 2 | — | |
RKDUDJILSVKJSN
|
7.4 | IC50 | 2 | — | |
YATBPBJXOBLSKJ
|
7.4 | IC50 | 2 | — | |
SXDFJZINGTYEHU
|
7.4 | IC50 | 2 | — | |
WSPFOBDEROUNMO
|
7.4 | IC50 | 2 | — | |
HCONGYLPWCJLSG
|
7.4 | IC50 | 2 | — |