Target Details
| UniProt AC | Q9BUB5 |
|---|---|
| Gene Symbol | MKNK1 |
| Protein Name | MAP kinase-interacting serine/threonine-protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 445
- Clinical molecules 13
- Avg pChEMBL 7.24
KEGG Pathways (3)
Active Molecules (445)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OROGTVJVVOAHJX
|
8.3 | IC50 | 2 | — | |
OROGTVJVVOAHJX
|
8.3 | IC50 | 2 | — | |
PBFMGCZSHKQYOU
|
8.2 | IC50 | 2 | — | |
NFYSHFWLDDXPKM
|
8.2 | IC50 | 3 | — | |
PNJVSKGBROJKNX
|
8.2 | IC50 | 2 | — | |
KKBIMZUEOUDERI
|
8.2 | IC50 | 2 | — | |
GXGBEOFIFZVLQU
|
8.2 | IC50 | 2 | — | |
PYHRNXAACBOPCP
|
8.2 | IC50 | 3 | — | |
LVSWSCZOVNFBCZ
|
8.2 | IC50 | 3 | — | |
GQAOHVZJKCGBQW
|
8.2 | IC50 | 2 | — | |
LWTZXHOFUFUYRH
|
8.2 | IC50 | 2 | — | |
JIBSLIWLWMKJGN
|
8.2 | IC50 | 3 | — | |
JTIWPTIGAVIWDG
|
8.2 | IC50 | 2 | — | |
GXOJOLCVOSVXPG
|
8.2 | IC50 | 3 | — | |
MPUZHXLKCBEGNC
|
8.2 | IC50 | 2 | — | |
TVPNRZPKPMXWJO
|
8.2 | IC50 | 2 | — | |
QSNAMJCLIIQNPP
|
8.1 | IC50 | 2 | — | |
GLKYGVDXWJUOFW
|
8.1 | IC50 | 3 | — | |
CUBNJCCNGYAEDF
|
8.1 | IC50 | 2 | — | |
BIBRQIOPTKIPOZ
|
8.1 | IC50 | 2 | — | |
VPJLAZUHVNGPLW
|
8.1 | IC50 | 2 | — | |
VENBOQULCZPZRI
|
8.1 | IC50 | 2 | — | |
KGLJXZUKNYLHMK
|
8.1 | IC50 | 2 | — | |
LZWVSDSGWLASHL
|
8.0 | IC50 | 2 | — | |
RKNGTCDEHZFRSK
|
8.0 | IC50 | 2 | — | |
CXNIDEGZWPEOCF
|
8.0 | IC50 | 3 | — | |
PXKYYYJETYKSIZ
|
8.0 | IC50 | 2 | — | |
DTEWSDGBCMIPIZ
|
8.0 | IC50 | 2 | — | |
XHBVYDAKJHETMP
|
8.0 | IC50 | 24 | Yes | |
YQVUADHJKWJHAF
|
8.0 | IC50 | 2 | — | |
QZAPGJZGBUIRLB
|
7.9 | IC50 | 2 | — | |
FMGALEFRCKPSHT
|
7.9 | IC50 | 2 | — | |
DUHHTOOYELYHTE
|
7.9 | IC50 | 2 | — | |
KXZLWAAQYGMLJX
|
7.9 | IC50 | 3 | — | |
ZMKWRVSEWQLUIX
|
7.9 | IC50 | 2 | — | |
VCRXHIDEBJOEFB
|
7.9 | IC50 | 2 | — | |
DFEIRHDGCVPKOC
|
7.8 | IC50 | 2 | — | |
QWBPEPMXXPKLGH
|
7.8 | IC50 | 2 | — | |
DJPQIFRWWIYXCH
|
7.8 | IC50 | 2 | — | |
BBQVZHIHIVJRIC
|
7.8 | IC50 | 2 | — | |
RAVMZMGTHHJIMD
|
7.8 | IC50 | 2 | — | |
JTIWPTIGAVIWDG
|
7.8 | IC50 | 2 | — | |
NTLQCWXRQTUIRI
|
7.8 | IC50 | 2 | — | |
UWKJXDSZQTXARH
|
7.8 | IC50 | 2 | — | |
VDNGCTAWOOSJIU
|
7.8 | IC50 | 2 | — | |
KECYTGQDOMZAAR
|
7.8 | IC50 | 2 | — | |
CYVKSJTVMXLBEL
|
7.7 | IC50 | 2 | — | |
VPIDNMQLFOKKCY
|
7.7 | IC50 | 2 | — | |
XCQQKYFEUUGRAR
|
7.7 | IC50 | 2 | — | |
FNHGPHDXAKOIJJ
|
7.7 | IC50 | 2 | — |