Target Details
| UniProt AC | Q9BRS2 |
|---|---|
| Gene Symbol | RIOK1 |
| Protein Name | Serine/threonine-protein kinase RIO1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01163 (RIO1) |
Summary
- Multi-target molecules 15
- Clinical molecules 7
- Avg pChEMBL 6.84
KEGG Pathways (1)
Active Molecules (15)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UIARLYUEJFELEN
|
8.1 | Kd | 289 | Yes | |
XZXHXSATPCNXJR
|
7.6 | Kd | 165 | Yes | |
WINHZLLDWRZWRT
|
7.5 | Kd | 201 | Yes | |
YYLKKYCXAOBSRM
|
7.3 | Kd | 191 | — | |
UCBIQZUJJSVQHL
|
7.1 | Kd | 8 | — | |
JOOXLOJCABQBSG
|
7.0 | Kd | 139 | — | |
HKSZLNNOFSGOKW
|
6.9 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
6.9 | Kd | 213 | — | |
NHHQJBCNYHBUSI
|
6.5 | Kd | 220 | — | |
GCIKSSRWRFVXBI
|
6.4 | Kd | 109 | Yes | |
PIQCTGMSNWUMAF
|
6.4 | Kd | 137 | Yes | |
OYONTEXKYJZFHA
|
6.3 | Kd | 69 | Yes | |
CTNPALGJUAXMMC
|
6.2 | Kd | 151 | — | |
BPNUQXPIQBZCMR
|
6.2 | Kd | 83 | Yes | |
ZCBUQCWBWNUWSU
|
6.1 | Kd | 59 | — |