Target Details
| UniProt AC | Q9BQI3 |
|---|---|
| Gene Symbol | EIF2AK1 |
| Protein Name | Eukaryotic translation initiation factor 2-alpha kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF22949 (HRI2_3H) PF00069 (Pkinase) |
Summary
- Multi-target molecules 18
- Clinical molecules 2
- Avg pChEMBL 6.41
Associated Diseases (1)
Active Molecules (18)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
APPXQUDJLJXULP
|
7.6 | IC50 | 47 | — | |
QAEKSWBVYBVLNO
|
7.4 | IC50 | 5 | — | |
HFOKVVVCWLIUBP
|
7.2 | IC50 | 3 | — | |
VRQMAABPASPXMW
|
6.8 | Kd | 10 | — | |
KWZXRCBCAYLKPI
|
6.7 | IC50 | 3 | — | |
XUZMWHLSFXCVMG
|
6.5 | Kd | 24 | — | |
SIXVRXARNAVBTC
|
6.4 | IC50 | 12 | — | |
PRWSIEBRGXYXAJ
|
6.3 | IC50 | 4 | — | |
UBPYILGKFZZVDX
|
6.2 | Kd | 130 | Yes | |
WVXNSAVVKYZVOE
|
6.2 | Kd | 92 | — | |
BIIVYFLTOXDAOV
|
6.1 | Kd | 82 | Yes | |
BFSMGDJOXZAERB
|
6.0 | Kd | 33 | — | |
CXQHYVUVSFXTMY
|
6.0 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.0 | Kd | 149 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JOOXLOJCABQBSG
|
6.0 | Kd | 139 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |