Target Details
| UniProt AC | Q9BPZ7 |
|---|---|
| Gene Symbol | MAPKAP1 |
| Protein Name | Target of rapamycin complex 2 subunit MAPKAP1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF16978 (CRIM) PF25322 (RBD_SIN1) PF05422 (SIN1) PF16979 (SIN1_PH) |
Summary
- Multi-target molecules 106
- Clinical molecules 2
- Avg pChEMBL 7.32
KEGG Pathways (1)
Active Molecules (106)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CGBJSGAELGCMKE
|
9.5 | Ki | 11 | — | |
AJJYRWYJJMMKIT
|
9.0 | IC50 | 5 | — | |
JUVAOVBSTMBYPN
|
9.0 | IC50 | 5 | — | |
PZLDVTRVPWMLFG
|
9.0 | IC50 | 5 | — | |
HGZCDZAZJVNMKO
|
8.9 | IC50 | 5 | — | |
CVMZRJQIEUQWJM
|
8.8 | IC50 | 5 | — | |
JGRISWOXHZGZPV
|
8.7 | IC50 | 5 | — | |
SRNMUDAJXGNOIO
|
8.6 | IC50 | 5 | — | |
IRCGXDFJTQYSNR
|
8.6 | IC50 | 5 | — | |
KVLFRAWTRWDEDF
|
8.6 | IC50 | 5 | — | |
YTOAJUIMCNAYNE
|
8.6 | IC50 | 5 | — | |
AWOSFEUBLOFLFP
|
8.3 | IC50 | 6 | — | |
GYLDXIAOMVERTK
|
8.3 | IC50 | 9 | — | |
IMXHGCRIEAKIBU
|
8.3 | IC50 | 5 | — | |
QRKKQWDDVIUFBU
|
8.3 | IC50 | 4 | — | |
XGKILEKRCLGRHL
|
8.2 | IC50 | 5 | — | |
YZESSOQLEODPGP
|
8.2 | IC50 | 5 | — | |
UXCAKZGNKOZXBM
|
8.2 | IC50 | 7 | — | |
ZSIRAWAQTMHYAU
|
8.2 | IC50 | 4 | — | |
GBZWWXBLAZUCRP
|
8.1 | IC50 | 5 | — | |
ZSIRAWAQTMHYAU
|
8.1 | IC50 | 5 | — | |
RFSMUFRPPYDYRD
|
8.0 | IC50 | 5 | — | |
HGZOUPKZPOAOOQ
|
8.0 | IC50 | 6 | — | |
UUWNQXUHQXRBNH
|
7.9 | IC50 | 5 | — | |
BYZCGCXGJTYMTH
|
7.9 | IC50 | 4 | — | |
OYXPDKVBMCFEJF
|
7.9 | IC50 | 5 | — | |
OYXPDKVBMCFEJF
|
7.8 | IC50 | 4 | — | |
IZLPVLBNRGPOHA
|
7.8 | IC50 | 5 | — | |
CEPOCJCCKQHPAE
|
7.8 | IC50 | 5 | — | |
HGLCMJBIRQLJPN
|
7.8 | IC50 | 4 | — | |
VZVYLEDIUUZTCW
|
7.8 | IC50 | 6 | — | |
BYZCGCXGJTYMTH
|
7.8 | IC50 | 4 | — | |
RGOBXIPHRILFRR
|
7.7 | IC50 | 5 | — | |
YDFGZXSSYDSJRM
|
7.7 | IC50 | 6 | — | |
ZTBJFQZREBPBTH
|
7.7 | IC50 | 4 | — | |
KDPPBJICLACJMM
|
7.6 | IC50 | 4 | — | |
FRQVRSOKGHVPMC
|
7.5 | IC50 | 4 | — | |
BSJSHEXWIGDLOO
|
7.5 | IC50 | 6 | — | |
QSUSKMROELIXNC
|
7.4 | IC50 | 5 | — | |
FFGUSRSMWFYKGK
|
7.4 | IC50 | 5 | — | |
IZCQVAPJLOTNAA
|
7.4 | IC50 | 4 | — | |
MLNSAGOBCFMEKI
|
7.3 | IC50 | 6 | — | |
PQWPFGHFJVFZRW
|
7.3 | IC50 | 4 | — | |
NBOWVAHSFAXGLP
|
7.3 | IC50 | 4 | — | |
CSLVGODBTQVCKU
|
7.3 | IC50 | 5 | — | |
DMJNPFVKLJNTLB
|
7.3 | IC50 | 4 | — | |
UZDWSTIRHOFWOF
|
7.2 | IC50 | 4 | — | |
BJEPBULKEVIYBP
|
7.2 | IC50 | 6 | — | |
GIJFXKSWQBHECT
|
7.2 | IC50 | 4 | — | |
YWWPYXNVIYKBAB
|
7.2 | IC50 | 4 | — |