Target Details
| UniProt AC | Q9BJF5 |
|---|---|
| Gene Symbol | CDPK1 |
| Protein Name | non-specific serine/threonine protein kinase |
| Organism | Toxoplasma gondii |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF13499 (EF-hand_7) PF00069 (Pkinase) |
Summary
- Multi-target molecules 250
- Clinical molecules 4
- Avg pChEMBL 7.84
Active Molecules (250)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QBINFJIYMSCWHV
|
7.2 | IC50 | 3 | — | |
NNQNLIXHDLUEKW
|
7.2 | IC50 | 2 | — | |
YRYOEVHVROHLKR
|
7.2 | IC50 | 3 | — | |
ORXPWRFCRDSKTB
|
7.2 | IC50 | 2 | — | |
ALFCMIDACCFSPY
|
7.1 | IC50 | 2 | — | |
ZBMXRMRKJLDZCX
|
7.1 | IC50 | 2 | — | |
OWAHNIJXSIARTN
|
7.1 | IC50 | 2 | — | |
QRQNLTAPCVSPJM
|
7.1 | IC50 | 2 | — | |
BERSUAQTWMUYMU
|
7.0 | IC50 | 3 | — | |
OYZYYVWBGXJDCM
|
7.0 | IC50 | 3 | — | |
FQZWNMKPWCGUSW
|
7.0 | IC50 | 2 | — | |
RQWDDVSBYNIPPF
|
7.0 | IC50 | 2 | — | |
FLROVNJZAHFSEL
|
7.0 | IC50 | 2 | — | |
XNLZFVQIZBXQNM
|
7.0 | IC50 | 3 | — | |
GHQHPTZESKRASB
|
7.0 | IC50 | 3 | — | |
LZLHBIZNXYYRCT
|
7.0 | IC50 | 2 | — | |
POLUTDHHFRXNTH
|
7.0 | IC50 | 2 | — | |
DAIRRUAQSVPBCD
|
6.9 | IC50 | 2 | — | |
GKDGNKRGOJPYMM
|
6.9 | IC50 | 2 | — | |
YJRWKOLRMSYZHE
|
6.9 | IC50 | 3 | — | |
QFGDRGRJMYSRIW
|
6.9 | IC50 | 3 | — | |
RMKJKBCWXWSHSS
|
6.9 | IC50 | 2 | — | |
VZHQCVYEVMECQT
|
6.9 | IC50 | 2 | — | |
VPLRUYIVHZQYCE
|
6.9 | IC50 | 3 | — | |
RYTHFKJTOHUIJB
|
6.9 | IC50 | 3 | — | |
QAWHVZMZNTYGPK
|
6.8 | IC50 | 3 | — | |
QKWPGKWGXYCSIM
|
6.8 | IC50 | 3 | — | |
XFIGCAVKRPQHIW
|
6.8 | IC50 | 2 | — | |
YJNHTFUUPURWMM
|
6.8 | IC50 | 2 | — | |
CSXKZYFDPBVVPL
|
6.8 | IC50 | 2 | — | |
LMVAHLFZGWUGNF
|
6.7 | IC50 | 8 | Yes | |
LSPQVFVCYDZDQE
|
6.7 | IC50 | 2 | — | |
JERUHDOQWVDHGI
|
6.7 | IC50 | 2 | — | |
MCKMGYSAHQYEDC
|
6.7 | IC50 | 3 | — | |
TYGCWIRHRMMCNF
|
6.7 | IC50 | 3 | — | |
YMNGGNWWZGVESF
|
6.7 | IC50 | 2 | — | |
JFMDHVAWBLYOTK
|
6.7 | IC50 | 2 | — | |
QYQQAFASPRPEFS
|
6.6 | IC50 | 2 | — | |
PFDOYRBDNTWQJP
|
6.5 | IC50 | 2 | — | |
QVMWSFYCPYOKBR
|
6.5 | IC50 | 3 | — | |
BVPMUIYAHGRSDO
|
6.5 | IC50 | 2 | — | |
WNGTZCAFSHVKDM
|
6.4 | IC50 | 2 | — | |
JBBMCVYXSKRHOX
|
6.3 | IC50 | 2 | — | |
TZDJIUGMUUUAQD
|
6.3 | IC50 | 3 | — | |
IXORERCONFMYQK
|
6.2 | IC50 | 3 | — | |
DJAZYXTUKHPMNT
|
6.2 | IC50 | 3 | — | |
NJUDGLGIRWPONB
|
6.1 | IC50 | 2 | — | |
ZGFXAJBFDCMHTM
|
6.0 | IC50 | 3 | Yes | |
LXVCVZIBEYVACX
|
6.0 | IC50 | 2 | — | |
RBMYSNNHZNAYPK
|
6.0 | IC50 | 2 | — |