Target Details
| UniProt AC | Q9BJF5 |
|---|---|
| Gene Symbol | CDPK1 |
| Protein Name | non-specific serine/threonine protein kinase |
| Organism | Toxoplasma gondii |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF13499 (EF-hand_7) PF00069 (Pkinase) |
Summary
- Multi-target molecules 250
- Clinical molecules 4
- Avg pChEMBL 7.84
Active Molecules (250)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IIWIRJIDPJDBPK
|
7.8 | IC50 | 2 | — | |
CQFGWDHRGPACPU
|
7.7 | IC50 | 2 | — | |
IOMXIVABWISZJT
|
7.7 | IC50 | 3 | — | |
XDQVOICHYGWNLW
|
7.7 | IC50 | 2 | — | |
JRLNZLOGPPLOOP
|
7.7 | IC50 | 2 | — | |
UESYKRUJFLCOLW
|
7.7 | IC50 | 5 | — | |
KMHCRQINFJTBPW
|
7.7 | IC50 | 2 | — | |
QXIVTEDEXTWOOT
|
7.7 | IC50 | 2 | — | |
WNSGCGVEGBFXSZ
|
7.7 | IC50 | 3 | — | |
AMFCAKSMRMMQBW
|
7.7 | IC50 | 2 | — | |
OZTUULYOGSAFBT
|
7.7 | IC50 | 3 | — | |
RWIWWMXAHPTNKT
|
7.7 | IC50 | 2 | — | |
IXXZPOFDZSFZBQ
|
7.7 | IC50 | 2 | — | |
SBQVLMWVGFDHFM
|
7.6 | IC50 | 2 | — | |
RXTBOWBIOOJHHA
|
7.6 | IC50 | 2 | — | |
GDQXJQSQYMMKRA
|
7.5 | IC50 | 15 | — | |
YJMHWCFTOAMRPN
|
7.5 | IC50 | 2 | — | |
GFAVGLXIXAHTSJ
|
7.5 | IC50 | 2 | — | |
GMXXNWXPTIGTFB
|
7.5 | IC50 | 2 | — | |
PLNJHRJUAXDDTJ
|
7.5 | IC50 | 2 | — | |
BJNUCAZGXXFVAJ
|
7.5 | IC50 | 2 | — | |
ALCIEJZDGYBETD
|
7.5 | IC50 | 2 | — | |
BAJCQXWKKBBHQY
|
7.5 | IC50 | 2 | — | |
WIEJOJTVAQUWEJ
|
7.5 | IC50 | 2 | — | |
WKSFPWSGPLXNBT
|
7.5 | IC50 | 2 | — | |
BSGWEWBSWAVORO
|
7.4 | IC50 | 5 | — | |
FCDBILPMWMBUOR
|
7.4 | IC50 | 2 | — | |
CJFWNLXLAAHQJY
|
7.4 | IC50 | 11 | Yes | |
BUYPQZTWWIVHDK
|
7.4 | IC50 | 2 | — | |
DUPSNQFPAJUAKA
|
7.4 | IC50 | 9 | Yes | |
KAEFKAWNHDHBCY
|
7.4 | IC50 | 3 | — | |
BNKSOMZUHDZTOZ
|
7.4 | IC50 | 2 | — | |
QCAIXILBXUUYFL
|
7.4 | IC50 | 2 | — | |
JEGPESWANUNSEW
|
7.4 | IC50 | 2 | — | |
PNBDCDXPQZPIPK
|
7.3 | IC50 | 3 | — | |
JHFJTTIYEGPPOW
|
7.3 | IC50 | 3 | — | |
OXQCNDDWRHBCGM
|
7.3 | IC50 | 2 | — | |
JXRWVEKMMXMIKO
|
7.3 | IC50 | 2 | — | |
XDITWQGWVWRWLJ
|
7.3 | IC50 | 2 | — | |
RZJSWJLAOYUVRB
|
7.3 | IC50 | 3 | — | |
YKVANMRHVMVLJX
|
7.3 | IC50 | 2 | — | |
YSPYRGQBCQIYBI
|
7.3 | IC50 | 2 | — | |
GVDYJBFFYVHNPA
|
7.3 | IC50 | 3 | — | |
CXUFYCPSBOYQMV
|
7.3 | IC50 | 5 | — | |
FWZKBBIJFGVHDF
|
7.3 | IC50 | 2 | — | |
YTTJKXSDNVYCBE
|
7.2 | IC50 | 3 | — | |
KGLWFPORHQPXJI
|
7.2 | IC50 | 3 | — | |
WZYJYIAEKIIPFR
|
7.2 | IC50 | 2 | — | |
XSHTUKYLKIKVFC
|
7.2 | IC50 | 2 | — | |
RGKPUWYSUXLERI
|
7.2 | IC50 | 3 | — |