Target Details
| UniProt AC | Q99986 |
|---|---|
| Gene Symbol | VRK1 |
| Protein Name | Serine/threonine-protein kinase VRK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 7
- Clinical molecules 1
- Avg pChEMBL 6.58
Associated Diseases (2)
Active Molecules (7)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DTEKTGDVSARYDS
|
7.5 | IC50 | 11 | — | |
AZJKTFMVKCDMSG
|
7.4 | Ki | 4 | — | |
DTEKTGDVSARYDS
|
7.0 | Ki | 3 | — | |
DSXXEELGXBCYNQ
|
6.1 | IC50 | 28 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |