Target Details
| UniProt AC | Q99928 |
|---|---|
| Gene Symbol | GABRG3 |
| Protein Name | Gamma-aminobutyric acid receptor subunit gamma-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 326
- Clinical molecules 0
- Avg pChEMBL 7.41
KEGG Pathways (7)
Active Molecules (326)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UFTKNTUWDMJOIX
|
8.4 | IC50 | 16 | — | |
UULFOYXSWNADTF
|
8.4 | IC50 | 16 | — | |
MKNXZRAKHYWDOS
|
8.4 | IC50 | 16 | — | |
XQUJTESAXUTXNH
|
8.4 | Ki | 16 | — | |
YGKSPOBIXHTPMV
|
8.3 | IC50 | 16 | — | |
ACMQMUZDLQDWTK
|
8.3 | Ki | 16 | — | |
GOCZPCXRIJMRNR
|
8.3 | Ki | 16 | — | |
PHOATQSOBKATTD
|
8.3 | Ki | 16 | — | |
PTRXPVDOTUGGHW
|
8.3 | IC50 | 16 | — | |
QWWODAPIEHJFQG
|
8.3 | IC50 | 16 | — | |
ZWWZTFYQCITUTK
|
8.3 | IC50 | 16 | — | |
BTLWEEGNXUJKKB
|
8.2 | IC50 | 16 | — | |
KIVQXKXZISOGBE
|
8.2 | Ki | 17 | — | |
NKIYALPHXLYICR
|
8.2 | IC50 | 16 | — | |
YUSWMAULDXZHPY
|
8.2 | Ki | 20 | — | |
ZRRVSALMQDOQAX
|
8.2 | Ki | 16 | — | |
BDISWVKOOATATE
|
8.2 | Ki | 16 | — | |
YUOOYQDBXTWPKL
|
8.2 | Ki | 16 | — | |
OTQXKRRISJPTFS
|
8.2 | IC50 | 16 | — | |
WMCJJXHYPNOCMT
|
8.2 | IC50 | 16 | — | |
ZRPUPUBWCXFOCY
|
8.2 | Ki | 16 | — | |
DKCAUMRZSZVJCP
|
8.1 | Ki | 16 | — | |
IVGTVZGLPHBTJV
|
8.1 | IC50 | 16 | — | |
IVGTVZGLPHBTJV
|
8.1 | IC50 | 16 | — | |
QVIQGNJPFOVZBZ
|
8.1 | Ki | 16 | — | |
YHNNMZUUFMJQQY
|
8.1 | IC50 | 16 | — | |
XGJLRKVQXMSBJW
|
8.1 | IC50 | 16 | — | |
KWPOKTUWXDCATM
|
8.0 | IC50 | 16 | — | |
AAOVKJBEBIDNHE
|
8.0 | IC50 | 16 | — | |
HQJSGBKPXYZTRN
|
8.0 | IC50 | 16 | — | |
MBZNSAJBODIJCK
|
8.0 | IC50 | 16 | — | |
PWFUHHSGSJDKCU
|
8.0 | IC50 | 16 | — | |
DVKHCFDZNVGRQT
|
8.0 | IC50 | 16 | — | |
HFPZDEHIDKJZSN
|
8.0 | Ki | 16 | — | |
LMJMBPXKXWIKQK
|
8.0 | IC50 | 16 | — | |
NNHRCSJWUBQYQV
|
8.0 | IC50 | 16 | — | |
PKJGSRHYDOGGLB
|
8.0 | Ki | 17 | — | |
ZJQHPWUVQPJPQT
|
8.0 | IC50 | 17 | — | |
FJLMOGVUSSSKEC
|
7.9 | Ki | 16 | — | |
LLAKESJIQFAQJA
|
7.9 | IC50 | 16 | — | |
CNVQMRWAJHEFGZ
|
7.9 | Ki | 16 | — | |
OPMIQGMTRGXAQY
|
7.9 | IC50 | 16 | — | |
VAARLVBAANTQOM
|
7.9 | Ki | 16 | — | |
HSEWUGOOPIEKBZ
|
7.9 | IC50 | 16 | — | |
XAMVDLCXXPEEEG
|
7.9 | Ki | 16 | — | |
YLRURIRIQRAQJJ
|
7.9 | Ki | 16 | — | |
WAEXHEOACCAOSS
|
7.8 | Ki | 16 | — | |
IMMPJABTWMVMPJ
|
7.8 | Ki | 16 | — | |
IQXJMMLNUIUGIQ
|
7.8 | Ki | 16 | — | |
PNRLOCDAUHBIHX
|
7.8 | IC50 | 16 | — |