Target Details
| UniProt AC | Q99873 |
|---|---|
| Gene Symbol | PRMT1 |
| Protein Name | Protein arginine N-methyltransferase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF13649 (Methyltransf_25) PF22528 (PRMT_C) |
Summary
- Multi-target molecules 86
- Clinical molecules 0
- Avg pChEMBL 7.3
KEGG Pathways (2)
Active Molecules (86)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SPEGERVLTUWZPA
|
8.5 | IC50 | 5 | — | |
BOGKHDNBFDMRMG
|
8.4 | IC50 | 3 | — | |
QTNIFNOIKLRHGJ
|
8.4 | IC50 | 2 | — | |
TXSFQHHRYLAEMB
|
8.4 | IC50 | 3 | — | |
WPAHUPFRZFNUKC
|
8.4 | IC50 | 2 | — | |
ICLYSKVLWUOLLZ
|
8.3 | IC50 | 2 | — | |
KJHBJSSYYMWKLQ
|
8.3 | IC50 | 3 | — | |
PMGPJYJFQITHHT
|
8.3 | IC50 | 3 | — | |
LIENDGUHQUTLMD
|
8.2 | IC50 | 3 | — | |
QVFVESAOLFEXQX
|
8.2 | IC50 | 3 | — | |
CNSBKLBZNFFFRD
|
8.1 | IC50 | 3 | — | |
AMPQIHZOWIDPQA
|
8.1 | IC50 | 2 | — | |
QTNIFNOIKLRHGJ
|
8.1 | IC50 | 2 | — | |
FMTVWAGUJRUAKE
|
8.0 | IC50 | 5 | — | |
FWIUJOSFDRYPNT
|
8.0 | IC50 | 2 | — | |
FUUQRIOHQLDOTR
|
8.0 | IC50 | 2 | — | |
AHBGFVBNHAXGOD
|
7.9 | IC50 | 3 | — | |
HHJFNFLLPHTDTH
|
7.9 | IC50 | 3 | — | |
GJDVMSRIXJKBKJ
|
7.8 | IC50 | 3 | — | |
QCPRDFJGTLMBCJ
|
7.8 | IC50 | 3 | — | |
ZKGHABBSYZLSAM
|
7.8 | IC50 | 2 | — | |
DYDJINHRKAERSQ
|
7.8 | IC50 | 2 | — | |
FYZDIUPNFFHKJM
|
7.8 | IC50 | 2 | — | |
NSMVLEXMOMOBHV
|
7.8 | IC50 | 2 | — | |
NSMVLEXMOMOBHV
|
7.8 | IC50 | 2 | — | |
DVZZYZNFLHFCPI
|
7.8 | IC50 | 7 | — | |
WJJPSVIYQWOSFK
|
7.7 | IC50 | 3 | — | |
UOYRGGRFVPHLEJ
|
7.6 | IC50 | 3 | — | |
MDBHVKTYIGBDLO
|
7.6 | IC50 | 3 | — | |
MOWUZOHGLGUMND
|
7.6 | IC50 | 2 | — | |
YDVOPOIVFHFPTA
|
7.5 | IC50 | 2 | — | |
LUBCTIQAZDQPJR
|
7.5 | IC50 | 5 | — | |
LTPABOINPMWTKU
|
7.5 | IC50 | 3 | — | |
PFNIKRLIXXKHOH
|
7.5 | IC50 | 2 | — | |
UXQWECXRONTUQW
|
7.4 | IC50 | 3 | — | |
QRXRBRDDXIISAI
|
7.4 | IC50 | 2 | — | |
XSOARJRAIKUXSE
|
7.4 | IC50 | 2 | — | |
YOCSLRCPVKLWMS
|
7.4 | IC50 | 3 | — | |
UOYQDRFGWGTDNI
|
7.3 | IC50 | 2 | — | |
LIVCXRSDQOQURR
|
7.3 | IC50 | 3 | — | |
MPASEZSHHLMDOX
|
7.3 | IC50 | 2 | — | |
ILHAASUEJBNZOF
|
7.3 | IC50 | 2 | — | |
CNMWTZSRTFSQJJ
|
7.2 | IC50 | 5 | — | |
MOPCOJLFDMFKCS
|
7.2 | IC50 | 4 | — | |
VYBORVUUKYMIGQ
|
7.2 | IC50 | 2 | — | |
KUAIUYDMQDZPEQ
|
7.2 | IC50 | 2 | — | |
KWRBLASCKRNYTH
|
7.2 | IC50 | 3 | — | |
DICKVPVLKDVBPQ
|
7.2 | IC50 | 3 | — | |
HDLMOUYGUDJTRP
|
7.2 | IC50 | 3 | — | |
SYRKWCSTKUNNAO
|
7.2 | IC50 | 2 | — |