Target Details
| UniProt AC | Q99814 |
|---|---|
| Gene Symbol | EPAS1 |
| Protein Name | Endothelial PAS domain-containing protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF23171 (bHLH_HIF1A) PF11413 (HIF-1) PF08778 (HIF-1a_CTAD) PF00989 (PAS) PF14598 (PAS_11) |
Summary
- Multi-target molecules 107
- Clinical molecules 0
- Avg pChEMBL 6.88
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (107)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FBCWKAJVKFDCBP
|
6.0 | IC50 | 2 | — | |
MEZFKPBDAMJHTJ
|
6.0 | IC50 | 2 | — | |
MKWIPRORQSLGLB
|
6.0 | IC50 | 2 | — | |
CIJFRPODNXMJFU
|
6.0 | IC50 | 2 | — | |
XQKWZFOJRRNGGD
|
6.0 | IC50 | 2 | — | |
FSJDOSKYUBIXLN
|
6.0 | IC50 | 2 | — | |
IWZDPCWOVHHKAW
|
6.0 | IC50 | 2 | — |